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2-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-methoxy-6-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}phenol
6-[3-(2-methoxyethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]quinoxaline
1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-2-(pyrrolidin-1-ylmethyl)piperidine
2,3-dimethyl-5-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
(2S)-2-amino-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}hexan-1-one
1-(cyclobutylmethyl)-3-hydroxy-3-{[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]methyl}piperidin-2-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
2-(3-methyl-4-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}-1H-pyrazol-1-yl)ethan-1-ol
2-{[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethan-1-ol
2-(2-chloro-4-fluorophenyl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(4-fluoro-3-methoxyphenyl)methyl]amine
N-benzyl{[1-(2-chlorophenyl)-5-oxopyrrolidin-3-yl]amino}sulfonamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-methoxy-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-ethyl-8-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-(2-methoxyphenyl)-1-(pyridine-4-carbonyl)pyrrolidine-3-carboxylic acid
2-{[(1-propylcyclobutyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-(1-phenylcyclopentyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-[(cyclopropylmethyl)amino]-N-(3,5-dimethoxyphenyl)-5-(dimethylsulfamoyl)benzamide
(1S,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
6-cyclopropyl-N-[(5-methoxy-1H-indol-2-yl)methyl]pyrimidin-4-amine
[(3R,4R)-1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-phenylpyrrolidin-3-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-{[3-(4-chlorophenyl)piperidin-1-yl]methyl}-N-ethylpyrimidin-2-amine
1-{[7-chloro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
(3S,4S)-N-[3-(3-fluorophenyl)phenyl]-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
2-ethyl-9-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-[2-amino-4-(trifluoromethyl)pyrimidine-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(cyclopent-3-en-1-yl)-7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-methoxyphenyl)-4-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
4-{[(1R,5S,6R)-3-(2-methylbenzoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}piperazin-2-one
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
3-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-{4-[2-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]phenyl}acetamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(3-hydroxy-2,2-dimethylpropyl)-1,3-oxazole-4-carboxamide
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoxaline-6-carboxamide
6-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]quinoline
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
3-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
ethyl 4-[2-(1H-imidazol-2-yl)benzoyl]piperazine-1-carboxylate
4-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-1-methyl-2-phenylpiperazine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-phenylpyridazin-3-amine
N-cyclohexyl-3-{4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propanamide
6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one