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[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
2-[1-(3-phenylpropyl)-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-[2-(1H-pyrazol-1-yl)ethyl]-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
5-methyl-N-[2-(morpholin-4-yl)ethyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(3-fluorophenyl)-3-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
[3-(2-phenylethyl)-1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl]methanol
2-(3-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenoxy)acetamide
(4aS,7aR)-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
8-[(3,5-difluorophenyl)methyl]-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(dimethyl-1,2-oxazol-4-yl)-3-hydroxypiperidine-1-carboxamide
methyl 3-[(4-ethoxyphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2,4-dimethoxyphenyl)-2-(methylamino)pyridine-3-carboxamide
7-fluoro-3-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
(3-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)urea
methyl 1-[(3R,5S)-1-[(2-ethoxyphenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)acetic acid
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-fluoro-1H-1,3-benzodiazole
1-{imidazo[1,2-b]pyridazin-6-yl}-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazine
2-[4-(pyrimidin-2-yloxy)phenyl]-1H-1,3-benzodiazole-5-carbonitrile
ethyl 1-(5-benzamido-1-cyclopentyl-1H-1,3-benzodiazole-7-carbonyl)piperidine-3-carboxylate
3-[2-({[2-(1H-imidazol-1-yl)propyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[2-(diethylamino)ethyl]methylamine
N-(1-cyclohexanecarbonylazepan-3-yl)cyclopropanecarboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
methyl (1R,3S,3aR,6aS)-5-benzyl-3-(3-cyanophenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[1-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
2-{1-[(5-cyclohexylthiophen-2-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
6-methyl-2-[(1-methylpiperidin-4-yl)amino]pyridine-3-carbonitrile
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[2-(thiophen-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-5-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
8-fluoro-3-[2-hydroxy-2-(pyridin-3-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-benzyl-2-(4-{4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
2-(2-methoxyethyl)-9-(6-methyl-2-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(pyridin-3-yl)acetyl]-1,4-diazepan-5-one
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanamide
2-amino-4-{[(1R)-2-hydroxy-1-phenylethyl]amino}quinazoline-6-carboxylic acid
{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
5-cyclobutyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
2-methoxy-3-(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
1-(9H-fluoren-2-ylmethyl)-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-acetyl-8-(3,4-dimethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane