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6-methyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
3-[(2-fluorophenyl)formamido]-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)propanamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-amino-6-(pyridin-3-yl)-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
3-({4-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]pyrimidin-2-yl}(methyl)amino)-N-methylpropanamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}azocane
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2,5-dimethylphenyl)-3-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)propanamide
N-{4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanamido]-2-methoxyphenyl}-3-methylbutanamide
4-(furan-3-yl)-N,6-dimethyl-2-oxo-N-(quinolin-6-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(3aS,6aS)-N-(2,3-dichlorophenyl)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
1-{[1-(2,3-dimethylphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
methyl 6-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridine-3-carboxylate
(3S,9aR)-3-benzyl-2-methyl-8-[(3-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-(cyclohexylmethyl)-4-[(dimethylsulfamoyl)amino]pyrrolidin-2-one
ethyl 4-(2-phenoxyethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylate
2-phenoxy-1-[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]ethan-1-one
1-methyl-2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-dihydroquinoline-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-4-methylpyrimidine-5-carboxamide
4-[3-(ethoxymethyl)-4-methoxyphenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[2-(1-ethyl-1H-pyrazol-4-yl)-7-methylquinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
4-(4-methylphenoxy)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
4-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
4-[(3-methylphenyl)methyl]-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[cyclopentyl(prop-2-en-1-yl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
N-(2-chlorophenyl)-3-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}propanamide
2-oxo-8-(4-propylpyrimidine-5-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl (2S,4S)-4-(2-cyclopropylquinoline-4-amido)-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxylate
2-fluoro-N-methyl-5-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]carbamoyl}amino)benzamide
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
4-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carbonyl}morpholine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3,4-trimethoxybenzamide
1,3-dimethyl-N-[1-(2-methylphenyl)cyclopropyl]-1H-indole-2-carboxamide
1-[1-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperidin-4-yl]piperidin-4-ol
9-(5-chloro-2-hydroxybenzoyl)-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
ethyl 2-[(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetate
1-(3-chlorophenyl)-4-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}piperazine
N3-ethyl-N5-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
3-(2-acetylphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-{[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}propane-1,2-diol
6-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
2-(4-fluoro-3-methylphenyl)-2-{methyl[4-(morpholin-4-yl)butyl]amino}acetic acid
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-methyl-6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-2-amine
8-{2-[methyl(propan-2-yl)amino]acetyl}-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-6-hydroxy-1,4-diazepan-1-yl}pyridine-3-carbonitrile