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(3S,4S)-1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrrolidin-3-ol
N-[2-(3-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenoxy)propyl]-5-methylthiophene-2-carboxamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
3-{[1-(4-carbamoyl-1,3-thiazol-2-yl)piperidin-4-yl]methyl}benzoic acid
3-(4-methyl-1,3-thiazol-5-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
3-[(dimethylamino)methyl]-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-ol
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,4,4-trifluorobutanamide
1-[3-(methoxymethyl)pyrrolidin-1-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
N-({7-[1-(4-chlorophenyl)cyclopropanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
8-(5-hydroxypyrazine-2-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3-{[1-(1,4-dithiepan-6-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(2-methoxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
7-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
2-cyclopropyl-N,4-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
9-(2,3-dimethyl-1H-indole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1S,5R)-6-(cyclobutylmethyl)-3-(pyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-amino-6-{4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-1-yl}pyrimidin-4-ol
4-[(2,2-difluoroethyl)sulfamoyl]-N-[2-(1H-pyrrol-1-yl)ethyl]benzamide
(3E)-N-{[1-(quinolin-8-ylmethyl)pyrrolidin-3-yl]methyl}pent-3-enamide
N-{1-[1-(8-fluoroquinoline-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-[(1S,2R)-2-aminocyclobutyl]-1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethylazepane-2-carboxamide
[(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(dimethylamino)pyrrolidin-2-yl]methanol
6-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-9H-purine
2-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-{3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[1-(piperidin-1-yl)ethyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]furan-2-carboxamide
2-(2-chlorophenyl)-N-(2,2-difluoroethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(4S)-3,3,4-trimethyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-ol
(butan-2-yl)({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amine
4-(1-methyl-1H-pyrazole-5-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
3-(3-fluorophenyl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methyl-N-(2-methylphenyl)piperidine-1-carboxamide
1-methyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-[2-(2,1,3-benzoxadiazol-5-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
2-[4-(propan-2-yl)morpholin-2-yl]-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
7-(isoquinoline-5-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-(4-aminopyrimidin-2-yl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
2-hydroxy-3-methyl-N-[3-(pyridin-3-yl)propyl]benzamide
N-(3-phenylprop-2-yn-1-yl)-N-propyl-4-sulfamoylbenzamide
[(2-methyl-1H-imidazol-4-yl)methyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[3-(dimethylamino)propyl]acetamide
3-[2-(dimethylamino)ethyl]-1-(6-methoxyquinolin-8-yl)-3-(oxolan-2-ylmethyl)urea
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-4-ethylpiperidin-4-yl]methanol
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-butyl-3-(2-hydroxyphenyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
2-[2-(dimethylamino)ethyl]-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one