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4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1-phenylbutan-1-one
4-(4-methoxyphenyl)-3-(1H-pyrazol-4-yl)-4H-1,2,4-triazole
(1R,2R,6S,7S)-N-(3,4-dimethylphenyl)-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
3-{[4-(4,6-dimethoxypyrimidin-2-yl)piperazin-1-yl]methyl}benzonitrile
3-(furan-2-yl)-2-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]propan-1-ol
1-[5-(3-benzyl-1H-1,2,4-triazol-5-yl)-2-methylphenyl]imidazolidin-2-one
[(3aS,6aS)-2-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-{[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
5-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(morpholin-4-yl)pyrimidin-2-amine
N-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanesulfonamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl (1S,3S,3aR,6aS)-5-ethyl-3-(4-fluoro-2-methoxyphenyl)-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
N-(1H-1,3-benzodiazol-2-yl)-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]acetamide
(3R,7S,8aS)-7-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-[(2-aminopyridin-3-yl)methyl]piperazine-2-carboxylic acid
N-{[3-(pyridin-3-yl)-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl]methyl}acetamide
2-{4-[(2E)-4-methylpent-2-en-1-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(2-butyl-1H-imidazol-4-yl)methyl]-2-(4-fluorophenyl)piperidine
4-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
(2S,4R)-4-amino-1-[3-(3,4-dimethylphenyl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
2-(2-fluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-chloro-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-(1H-pyrazol-1-yl)benzamide
2-{4-methyl-6-[(oxan-4-yl)amino]pyrimidin-2-yl}phenol
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(4-phenylbutyl)acetamide
2-({6-[(1-cycloheptylpiperidin-3-yl)amino]pyrimidin-4-yl}amino)ethan-1-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(piperidin-4-yl)amino]pyridine-3-carboxamide
N-benzyl-N-ethyl-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
9-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopentyl-9-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]pyrimidin-4-amine
4-{4-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(2-methoxyphenyl)methyl](pyridin-4-ylmethyl)amine
N-ethyl-1,3-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-methyl-5-propyl-1-benzofuran-2-carboxylic acid
N-[2-(1H-pyrrol-1-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-(cyclopropylmethyl)-5-[(4-acetamidophenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{[(4-methoxy-3-methylphenyl)methyl]amino}-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxyethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})(1H-pyrazol-5-ylmethyl)amine
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-(1,3-thiazol-2-ylmethyl)urea
4-(2-phenylethyl)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
(3S,4S)-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol