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1-butyl-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
1-(1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}azetidin-3-yl)piperidine
4-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyrimidine
2-(pyridin-3-ylmethyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-N-ethylacetamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
N-[(4-methoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)oxolane-3-carboxamide
(4S)-3-{2-[4-(2-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
methyl 3-(2,5-dimethylfuran-3-carbonyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(5-{[4-(thian-4-yl)piperazin-1-yl]methyl}furan-2-yl)benzonitrile
methyl 4-({2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamido}methyl)benzoate
5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
3-(1-benzofuran-2-yl)-1-benzyl-4-(1H-imidazol-2-yl)-1H-pyrazole
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylphenyl)methyl]piperazine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]piperidine-3-carbonitrile
N-[3-(4-{[(1-hydroxycyclohexyl)methyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-({1-[(2R)-2-aminopropanoyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
3-[(3R,4S)-4-(dimethylamino)-1-{[2-(propan-2-yl)phenyl]carbamoyl}piperidin-3-yl]propanoic acid
5-[(3,5-dimethoxyphenyl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1S,5R)-6-(5-propylthiophene-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-cyclopentyl-N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
2-(1H-indazol-1-yl)-N-[(1-methylpiperidin-3-yl)methyl]acetamide
2-[methyl({4-methyl-5-[1-(pyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2,6-difluoro-4-methoxy-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
4-[(2,3-difluorophenyl)methyl]-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
methyl 3-(3-methoxybenzamido)-5-{[3-(pyridin-3-yl)propanamido]methyl}benzoate
diethyl({[2-(1-ethylpiperidin-3-yl)ethyl]sulfamoyl})amine
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
1-(1-cyclopropanecarbonylpiperidine-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
[(5-ethylpyridin-2-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}propanamide
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-4,4,4-trifluorobutanamide
N-cyclopentyl-6-[3-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-ethylpyrimidine
2-amino-4-(3-chloro-4-methoxyphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
(2,2-diphenylethyl)(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(pyrrolidin-1-ylmethyl)pyridine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-2-yl]methanesulfonamide
1-[2-(4-fluorophenyl)azetidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
methyl 4-{4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperazin-1-yl}benzoate
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(thiophen-2-yl)ethyl]pyrrolidin-2-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(3,4-difluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-[(2,5-difluorophenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one