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N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)quinoline-6-carboxamide
N-(2-methylphenyl)-2-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}acetamide
4-benzyl-3-[1-(furan-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methyl-2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
(2R,3R)-3-amino-1'-[(2E)-3-phenylprop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-[3-(dimethylamino)pyrrolidin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[(2,4-dichlorophenyl)methyl]-3-(1-ethyl-1H-1,2,4-triazol-3-yl)urea
7-(cyclobutylmethyl)-2-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-fluoropyridine
N-(2,4-dimethoxyphenyl)-3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}propanamide
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]pyridine-4-carboxamide
4-(1H-pyrazol-1-yl)-1-[(thiophen-2-ylmethyl)carbamoyl]piperidine-4-carboxylic acid
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-chloro-N-[1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
7-cyclohexyl-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}-5-methoxyphenol
3-(1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-(2-methylfuran-3-carbonyl)-4-(3-methylphenoxy)piperidine
4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-1λ6-thiomorpholine-1,1-dione
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
[1-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxypyridine-3-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
3,7-dimethyl-8-[3-(propan-2-yloxy)phenyl]-2,3,6,7-tetrahydro-1H-purine-2,6-dione
(1R,7S)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(prop-2-en-1-yl)-N-(pyridin-4-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-(1-phenylcyclopropanecarbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-[5-(but-3-en-1-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
(3S,4S)-4-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-1-(4-methoxybenzoyl)pyrrolidin-3-ol
3-[4-fluoro-3-(hydroxymethyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
6-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
2-[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)(methyl)amino]-N-methylacetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N,1-dimethyl-6-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}thiophen-3-yl)methyl]piperidine
2-{[5-(1H-pyrazol-5-yl)-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[3-(2-methoxyethyl)-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl]acetic acid
2-[3-(oxan-4-yl)-5-(5-oxopyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(3aR,7aS)-2-[2-(1H-imidazol-2-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}acetamide
[(3-chlorophenyl)methyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
(2,1,3-benzoxadiazol-4-ylmethyl)({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
N-benzyl-1-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-indole-3-carboxamide
N-methyl-2-oxo-N-[3-(oxolan-2-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-methoxyphenyl)methyl]piperidine-3-carboxamide