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1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-amino-4-(1-ethenyl-1H-pyrazol-4-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
1-ethyl-N-[(3-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzoate
2-[(1S,5R)-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyridine-3-carbonitrile
4-{2-[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}phenol
4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazine-1-sulfonamide
2-[3-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)-1H-indol-1-yl]acetamide
1-cyclopropanecarbonyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(methoxymethyl)-N-[2-(2-phenoxyethoxy)phenyl]cyclobutane-1-carboxamide
N,N-diethyl-2-{[4-(1H-imidazol-2-ylmethyl)-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl]oxy}acetamide
N-(2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]morpholin-2-yl}ethyl)methanesulfonamide
N-methyl-4-[(1-methyl-2-oxopyrrolidin-3-yl)sulfamoyl]-N-(prop-2-en-1-yl)benzamide
N-(cyclohexylmethyl)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidine-1-carboxamide
5-methoxy-3-methyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-indole-2-carboxamide
6-(3-fluoro-4-methoxyphenyl)-N-(2,2,2-trifluoroethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-fluoro-4-(trifluoromethyl)phenyl]-3-methylurea
N-(1,1-dioxo-1λ6-thian-4-yl)-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide
8-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(1H-indol-2-ylmethyl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
4-(6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)thiomorpholine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetamide
5-(azocan-1-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
[(5-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
N-(4-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)acetamide
N-ethyl-2-[2-fluoro-3-(trifluoromethyl)phenyl]pyrimidin-4-amine
7-(3,6-dimethylpyrazin-2-yl)-4-(oxolane-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2,6-dimethylpyridin-4-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
3-{[4-(cyclopentylmethyl)piperazin-1-yl]methyl}-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
3-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
methyl (2R)-2-({1-[(2-methoxyphenyl)methyl]-5-[(3-methylbutyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}formamido)propanoate
(1R,3S)-7-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
3,5-dimethyl-1-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azetidin-3-yl)-1H-pyrazole
methyl 5-cyano-6-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-methylpyridine-3-carboxylate
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridine-3-carbonyl)-1,4-diazepan-5-one
[(2S,4R)-4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-methylpyrrolidin-2-yl]methanol
2-ethoxy-N-[1-(3-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]acetamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
3-[2-(4-methoxyphenyl)ethyl]-1-[(4-methyl-1,4-oxazepan-6-yl)methyl]urea
2,6-dimethyl-N-[2-(pyridin-3-ylformamido)ethyl]pyridine-4-carboxamide
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-methanesulfonylphenyl)-3-[3-(trimethyl-1H-pyrazol-1-yl)propyl]urea