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(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-(3-methoxypropyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
4-fluoro-N-{2-[(3-propyl-1H-pyrazol-5-yl)formamido]ethyl}benzamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(pent-4-enoyl)piperidine-3-carboxylate
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-phenyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]cyclohexane-1-carboxamide
1-methyl-N-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,5S,6R,7S)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2S)-N-[3-(3-methylphenyl)phenyl]-1-(1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-benzyl-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methoxy-N-{2-[4-(propan-2-yl)phenyl]phenyl}acetamide
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]quinoxaline-6-carboxamide
2-methyl-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-(1,2-oxazol-3-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
2-methyl-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
6-[(2R)-2-hydroxypropyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N,N-bis(2-hydroxyethyl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-ethyl-9-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-[(1-ethyl-1H-indol-6-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[3-ethyl-5-(4-methyl-2-phenylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-(1-ethyl-1H-pyrazol-4-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-[(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
5-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,6-dimethylthieno[2,3-d]pyrimidin-4-amine
5-chloro-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(methylsulfanyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-benzyl-2-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
3-(4-fluorophenyl)-N-(2-methoxyethyl)-N-propyl-1H-pyrazole-5-carboxamide
2-{2-[4-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-1-yl]ethoxy}ethan-1-ol
1-(2,5-dimethoxyphenyl)-2-(propan-2-yl)-1H-imidazole
4-(1,3-dihydroxypropan-2-yl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
1-{[(3R,4R)-4-(hydroxymethyl)-1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}pyrrolidin-3-yl]methyl}piperidin-4-ol
[1-(5,6-dimethylpyrimidin-4-yl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
2-(3-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}piperidin-1-yl)acetamide
{4-[(3-fluorophenyl)methyl]-1-(pyrimidin-2-yl)piperidin-4-yl}methanol
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]azepane
2-(2,5-dioxoimidazolidin-4-yl)-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}acetamide
(3S,4S)-1-{[(4-fluorophenyl)methyl]carbamoyl}-4-propylpyrrolidine-3-carboxylic acid
1-(4-amino-6,7-dimethoxyquinazolin-2-yl)-1,4-diazepan-6-ol
7-(4-chloro-1H-pyrazole-3-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(5-hydroxypyrazine-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-cyclopropyl-8-[(4-ethoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclobutanecarbonyl-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
8-[(4-hydroxyphenyl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-6,7-dimethyl-1H-1,3-benzodiazole
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
2-methyl-8-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-fluoro-4-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one