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2-{1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}-N-methylpropanamide
N-[(3S,4R)-4-propyl-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]acetamide
7-(2-methoxyethyl)-2-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(azepan-1-yl)ethyl]-N-methylacetamide
2-phenyl-7-phenylmethanesulfonyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aS,8aR)-1-propyl-6-(2-propyl-1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(furan-3-carbonyl)piperidine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4,4,4-trifluorobutanamide
2-(azepan-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
N-methyl-N-{2-phenyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]ethyl}thiophene-3-carboxamide
1-({[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]carbamoyl}methyl)piperidine-4-carboxamide
(3R,4R)-3-methyl-1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
2-amino-N-[(3-methoxyphenyl)methyl]-4-methyl-N-(2-methylpropyl)-1,3-thiazole-5-carboxamide
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-(azocan-1-yl)-1-[4-(4-hydroxybutyl)piperazin-1-yl]propan-1-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(2-chloro-4-fluorophenyl)-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}urea
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
ethyl 2-(1-{2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamido}cyclohexyl)acetate
5-{[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]carbamoyl}thiophene-2-carboxylic acid
4-{3-azaspiro[5.5]undecan-9-yl}piperazine-1-carboxamide
1-phenyl-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
2-(2,4-dioxoimidazolidin-1-yl)-N-{[(2-fluoro-4-methylphenyl)carbamoyl]methyl}acetamide
6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 1-(2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-[3-methyl-1-(pyridin-3-yl)butyl]urea
8-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazine-2-carboxamide
1-(2-phenylethyl)-4-[(2S)-1-(piperidin-4-yl)pyrrolidine-2-carbonyl]piperazine
2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-N-(furan-2-ylmethyl)acetamide
1-[(2,3-dimethoxyphenyl)methyl]-4-(oxan-4-yl)piperazine
10-methoxy-5-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-methylurea
(4aS,8aS)-2-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-decahydro-2,7-naphthyridin-4a-ol
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-N,N-bis(propan-2-yl)benzamide
methyl(1,2-oxazol-5-ylmethyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
1-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-[(4-methoxyphenyl)methyl]propanamide
1-(4,6-dimethoxypyrimidin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[3-(1H-pyrazol-5-yl)phenyl]-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxamide
ethyl 3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propanoate
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[7-(4-ethylpiperazine-1-carbonyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
6-(methoxymethyl)-1-methyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[(3-methoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(1,3-benzoxazol-2-ylmethyl)-1-(pyrimidin-2-yl)piperidin-4-amine