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1-(2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-[2-(ethylsulfanyl)ethyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
6-amino-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]pyridine-2-carboxamide
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
8-[(3,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
ethyl 2-[1-(3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperidin-2-yl]acetate
3-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-ol
2-(2-aminoethyl)-N,5,6-trimethyl-N-[3-(oxolan-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(3-phenylpropyl)-4-(pyridin-2-ylmethyl)morpholine
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
4-(4-{1-[2-(5-methylthiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
(2S,5R)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2,5-dimethylpiperazine
3-[2-(2-chlorophenoxy)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]piperidine-1-carboxylate
2-(1H-imidazol-1-yl)-N-[2-(2-phenoxyethoxy)phenyl]acetamide
N-({7-[2-(4-acetylphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
3-[(3R,4S)-1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(4aS,7aR)-1-(3-hydroxy-4-methylbenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[4-(dimethylcarbamoyl)phenyl]-4-ethoxybenzoic acid
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
N,2,3,5-tetramethyl-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-fluoro-5-methylphenyl)-N'-(prop-2-en-1-yl)-N'-(pyridin-3-ylmethyl)butanediamide
3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(4-methylphenyl)propan-1-ol
1-(4-methyl-1H-pyrrole-2-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-methoxy-1-{1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
4-(5-methylpyridin-2-yl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
(3R,5S)-N-butyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]piperidine-3-carboxamide
2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}thiophen-3-amine
2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
N-cyclopropyl-1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
3-(2-aminopyrimidin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
2-[(2-chlorophenyl)methyl]-4-{4-[(3,4-difluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
6-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(4-phenylbutan-2-yl)-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
3-{[1-(3,3,3-trifluoropropanesulfonyl)pyrrolidin-3-yl]methyl}benzamide
3-(morpholine-4-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methyl-1'-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-4-yl)propanamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
4-(4-hydroxy-3-methylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
N-[(1R,2S)-2-phenylcyclopropyl]-4-(1H-pyrazol-4-yl)butanamide
1-[4-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]ethan-1-one
(3S,4R)-1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(hydroxymethyl)piperidin-3-ol