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9-[(3,5-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(benzyloxy)-1-(2-methylpropyl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-2-one
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
6,6-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]pyrazin-2-ol
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
3-amino-1-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
N-methyl-5-{[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxyethan-1-one
7-chloro-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamido}ethyl)piperidine-3-carboxamide
N,N-dimethyl-5-[methyl(thiophen-2-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1R,5S)-6-methyl-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(pyridin-3-yl)piperazine
N-[1-(furan-2-carbonyl)piperidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
3-[(cycloheptylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(2-methylpropyl)amine
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-diethylacetamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-phenoxypropan-1-one
methyl (2R,4S)-1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-hydroxypiperidine-2-carboxylate
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
(3aR,6aS)-1-oxo-5-(4-phenylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(methoxymethyl)furan-2-carbonyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
4-{4-[(1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}-N-[(2-fluorophenyl)methyl]benzamide
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[3-(dimethylamino)propyl]-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-ethyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidin-2-one
6-chloro-2-(1H-pyrazol-3-yl)-1,3-benzothiazole
2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-methylphenyl)-5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyrimidin-4-ol
(3aS,6aS)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-4-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidine-1-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1'-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{[ethyl(oxan-4-yl)amino]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
1-{2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(2-methoxyphenyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridazin-3-amine
2-[benzyl(methyl)amino]-N-[(3-methylpyridin-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-cyclopentyl-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
1-[2-(N-methylmethanesulfonamido)ethyl]-5-oxopyrrolidine-3-carboxylic acid
N-[2-(4-fluorophenyl)ethyl]-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-3-methyl-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]quinoxaline-5-carboxamide
5-ethyl-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
1-[(4-fluorophenyl)methyl]-4-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-2-one
N-({1-[(2R)-2,3-dihydroxypropyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N,2,5-trimethylfuran-3-carboxamide