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1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-(4-fluorophenyl)-2-hydroxyethan-1-one
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
7-chloro-N-methyl-N-(2-methylpropyl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
2-[3-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methoxypyrimidine
2-(4-methoxyphenoxy)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(trifluoromethyl)pyrimidine
N-[2-(4-methylphenyl)propan-2-yl]piperidin-3-amine
1-cyclohexyl-N5-cyclopropyl-N3-methyl-4-oxo-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-(4-hydroxybutyl)-4-{[(4-methylphenyl)amino]methyl}benzamide
6-[3-(aminomethyl)pyrrolidin-1-yl]-2-(butylsulfanyl)pyrimidin-4-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(pyrazin-2-yl)acetyl]piperidin-3-yl}propanamide
N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}-3-propanamidobenzamide
7-chloro-N-(3-methyl-1,2,4-thiadiazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
3-[(cyclobutylcarbamoyl)methyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(4-chlorophenyl)-5-(1,4-dithiepan-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-cyclobutyl-2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetamide
1-(furan-2-ylmethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
7-fluoro-3-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzofuran-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[2-(diethylamino)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
3-(2-hydroxyphenyl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-cyclohexyl-3-(1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)benzamide
5-[(benzyloxy)methyl]-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
3-fluoro-2-(4-methanesulfonylphenyl)pyridine
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-1,2,3-thiadiazole-4-carboxamide
4-(1-ethyl-1H-pyrazole-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-1-yl}-1,3-benzothiazole
N,N-dimethyl-3-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
(2R)-2-({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanamide
N,N-dimethyl-4-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,3-thiazol-2-amine
(2S,4R)-4-amino-N-ethyl-1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
3-[5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1H-1,3-benzodiazol-1-yl]propan-1-ol
1-[(diethylcarbamoyl)methyl]-N-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-(1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}pyrrolidin-3-yl)acetamide
3-[5-(2-benzyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
N-methyl-N-[2-(morpholin-4-yl)propyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
4-{[1-(1-benzofuran-2-ylmethyl)piperidin-2-yl]methyl}morpholine
ethyl 1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
1-[1-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethyl]-4-methylpiperazine
(2S,4R)-4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]-N,N-diethylpyrrolidine-2-carboxamide