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6-ethyl-2-methoxy-3-{[(oxolan-3-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{4-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]piperidin-1-yl}ethan-1-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
methyl 4-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
N-(4-fluorophenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(5-ethylpyridin-2-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
7-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-oxa-7-azaspiro[4.5]decane
1-[2-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(1,3-thiazol-2-ylmethyl)amine
1-[(3-methylphenyl)methyl]-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,6-dimethylpyrimidin-4-amine
3-(4-hydroxyphenyl)-N-[3-(4-methoxyphenoxy)propyl]-N-methyl-1H-pyrazole-5-carboxamide
2-[2-(4-fluorophenyl)morpholine-4-carbonyl]-5-methoxy-1-methyl-1H-indole
8-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,6aR)-N,2-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(3aS,6aS)-2-[2-(1H-indazol-3-yl)acetyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
6-methyl-5-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}quinoline
5,7-dimethyl-N-[3-(methylsulfanyl)propyl]pyrido[2,3-d]pyrimidin-4-amine
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
N-(3-hydroxy-3-phenylpropyl)-1-[(4-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-({2-[1-(butane-1-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
N-(2-methoxyethyl)-1-methyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-1,3-benzodiazol-2-amine
2-(2-fluoro-5-methoxyphenyl)pyridine
2-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-6-(4H-1,2,4-triazol-4-yl)pyridine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(pyrazin-2-yl)propanamide
(2S,4S)-4-amino-N-ethyl-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]pyrrolidine-2-carboxamide
(1s,4s)-4-(4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-phenylethane-1,2-dione
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-{2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
5-{2-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
8-(1H-1,2,3-benzotriazole-5-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-({1-[(2S)-5-oxopyrrolidine-2-carbonyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
N-(2-{8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}thiophen-3-yl)acetamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-phenyl-1H-pyrazole-4-carboxamide
4,6-dimethyl-1-{2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
N-[4-(5-methylfuran-2-amido)phenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepan-5-one
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-(2-methylphenyl)propan-1-one
{3-[2-methoxy-6-(6-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]propyl}dimethylamine
6-oxo-N-[2-(pyridin-3-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-(2-{[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl)amino}ethyl)cyclopentan-1-ol
7-methyl-2-[2-methyl-2-(4-methylphenoxy)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2,4-difluorophenyl)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]acetamide