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2-(benzylsulfanyl)-N4-(pyridin-2-ylmethyl)pyrimidine-4,6-diamine
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)urea
3,7-dimethyl-11-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-3,7,11-triazaspiro[5.6]dodecane
7-fluoro-4-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-(2-{[7-(1H-imidazol-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)propanamide
2-chloro-6-fluoro-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-methylbenzamide
1-butyl-5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-3-methyl-1H-1,2,4-triazole
4,6-dimethyl-2-oxo-N-(2-propoxyethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-{1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-methanesulfonyl-N-methyl-N-(quinolin-4-ylmethyl)acetamide
N-(3-fluoro-4-methylphenyl)-4-(pyridin-4-yl)piperidine-1-carboxamide
N-ethyl-6-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-methylpyridazin-3-amine
6-cycloheptyl-3-ethyl-1-methyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{5-[(E)-2-phenylethenyl]-1H-indazol-1-yl}acetamide
1-(cyclopropylmethyl)-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3,4-difluorophenyl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
(2E)-3-(4-methoxyphenyl)-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)prop-2-en-1-one
3-[(3-propyl-1,2-oxazol-5-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
(3S,4S)-1-(2-amino-4-phenylpyrimidine-5-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3S,4S)-4-methyl-1-(1-phenylcyclohexanecarbonyl)piperidine-3,4-diol
4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methyl-1,3-oxazole
2-amino-6-tert-butyl-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-[4-(3-methoxypyridin-2-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-[2-(1-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
(3R,4S)-1-[2-(3-methylphenyl)benzoyl]-4-propylpyrrolidin-3-amine
3-(azepane-1-carbonyl)-N-[2-(4-methoxyphenyl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-(5-ethylthiophene-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-(piperidin-3-ylmethyl)benzamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxyacetamide
5-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-({5-cyclobutyl-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
methyl[(5-methylthiophen-2-yl)methyl]{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
2-(ethylsulfanyl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-[methyl(2-phenylethyl)amino]-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
1-acetyl-N-[2-(2-phenoxyphenyl)ethyl]piperidine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-{[2-(2-phenylethynyl)phenyl]methyl}pyrrolidine-2-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(4-methoxy-4-oxobutanoyl)piperidine-3-carboxylate
2-(2-methoxyethoxy)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
(1R,3S,5S)-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-ol
4-{4-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]phenyl}but-3-yn-1-ol
propan-2-yl 4-chloro-3-[2-(1H-imidazol-4-yl)acetamido]benzoate
N-(oxan-4-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide