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2-(cyclohex-1-en-1-yl)-1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
6-(2-aminoethyl)-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]pyrimidin-4-amine
2-{[(3S,4S)-4-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl]methyl}-8-fluoroquinolin-4-ol
[(3,4-dimethoxyphenyl)methyl](1,4-dioxan-2-ylmethyl)amine
1-cyclohexyl-N3-[(2-methoxyphenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(1-ethylpyrrolidine-3-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(1-phenylethyl)amine
methyl 1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidine-3-carboxylate
ethyl 4-[6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
5-ethyl-5-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)morpholine
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-ol
2-{5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}acetamide
1-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-amine
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}propanamide
(1R,7S)-3-cycloheptyl-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
(4aS,7aR)-1-(5-methoxyfuran-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,5-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(4-chlorophenyl)-5-(methanesulfonylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazole
2-methyl-5-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(4aR,8aR)-2-[(3-methyl-1H-indol-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
6-({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(4-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[(3S)-3-hydroxy-3-phenylpropyl]-3-methoxy-1,2-dihydropyridin-2-one
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
4-{[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
(2R,3R,6R)-5-(3-fluoropropyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(furan-3-carbonyl)-3-[2-methyl-3-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-[6-amino-5-cyano-4-(2-methoxy-3,5-dimethylphenyl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
4-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(thiophen-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-(2,4-dimethylpyrimidine-5-amido)piperidine-1-carboxylate
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-(furan-2-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2,7,8-trimethylquinoline-4-carboxamide
2-[2-(1H-imidazol-1-yl)ethyl]-N-(naphthalen-1-yl)piperidine-1-carboxamide