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3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
5-(1-benzyl-1H-pyrazole-4-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl (2S,4R)-4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3,4-dimethylphenyl)methyl]piperidin-3-ol
2-(4-fluorophenyl)-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]morpholine
4-(hydroxymethyl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-ol
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxoazepan-1-yl)acetamide
3-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-1λ6-thiolane-1,1-dione
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(2-methylprop-2-en-1-yl)benzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylacetamide
2-{1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-2-yl}pyridine
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
[(2,3-dimethyl-1H-indol-5-yl)methyl][(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-(6-methoxyquinolin-8-yl)-4-methyl-1,4-diazepane-1-carboxamide
3-[(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-4H-chromen-4-one
10-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
4-(hydroxymethyl)-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]piperidin-4-ol
(3S,4S)-1-[(2-methoxypyridin-3-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[(2-chlorophenyl)methyl]-N-(prop-2-yn-1-yl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-{2-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-{1-[(4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
(2S,4S)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-ethyl-N-phenyl-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
2-chloro-5-(5-{[3-(hydroxymethyl)piperidin-1-yl]methyl}furan-2-yl)benzoic acid
(2-methoxyethyl)({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
(3S,4R)-4-(2-methylphenyl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-3-carboxylic acid
{3-[(4-fluorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
4-[1-(3-ethoxypropanoyl)piperidin-3-yl]benzoic acid
1-cyclopropyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrrole-2-carboxamide
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
9-[(2S)-4-methyl-2-(methylamino)pentanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-methoxyethyl 3-methyl-3-phenylpiperidine-1-carboxylate
2-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,3-thiazole-4-carboxamide
6-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(1,4-dioxan-2-ylmethyl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
3-amino-1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
(3S)-3-ethyl-4-[4-methoxy-3-(morpholin-4-yl)benzoyl]morpholine
N-[4-(2-fluorophenoxy)phenyl]-1-(oxane-4-carbonyl)piperidine-4-carboxamide
1-{4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]phenyl}-1H-imidazole
6-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-methoxy-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide