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2-(4-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenoxy)acetic acid
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-methyl-2-(4-methylpiperazin-1-yl)-N-[2-(phenylsulfanyl)ethyl]pyrimidine-5-carboxamide
3-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-5-methyl-1,2-oxazole
1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
2-(4-chlorophenyl)-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
1-(cyclobutylmethyl)-3-hydroxy-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-(4-phenyl-1,2,3-thiadiazol-5-yl)piperidine-1-carboxamide
(3S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-[3-(dimethylamino)pyrazin-2-yl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
methyl 3-cyclohexaneamido-6-{[ethyl(pyridin-4-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
3-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-{1-[(4-fluorophenyl)methyl]-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl}acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl})amine
3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-[(3R,4S)-1-(5-fluoropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxylate
N-(3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
5-acetyl-3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
2-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-butyl-8-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-6-(pyrrolidin-1-yl)pyrimidine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[3-(methylsulfanyl)propyl]piperidine
[(2S)-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N,1-bis(propan-2-yl)-1H-pyrazole-3-carboxamide
4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane-1-carbaldehyde
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
2-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
2-(2,4-dichlorophenoxy)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-phenyl-1,4-diazepane-1-carboxamide
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
2-{1-[(4-methanesulfonylphenyl)methyl]pyrrolidin-3-yl}benzoic acid
N-[2-(dimethylamino)ethyl]-N-methyl-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
(2E)-N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(pyridin-4-yl)prop-2-enamide
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-N-{spiro[2.5]octan-1-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
ethyl 5-[(2S,4R,6S)-4-acetamido-6-(2-methylpropyl)oxan-2-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
dimethyl[2-(2-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
3-(5-{2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)-6-methylpyridazine
6-methyl-2-({methyl[1-(1,3-thiazol-5-yl)ethyl]amino}methyl)quinolin-4-ol