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N-[2-(3,5-dimethylphenoxy)ethyl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-methylacetamide
3-[5-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
2-[(2-methylphenyl)sulfanyl]-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
ethyl 4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazine
3-(1-ethyl-1H-imidazol-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(pyridin-4-yl)pyridine-3-carboxamide
N-[3-(cyclopentyloxy)propyl]-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
8-(6-methylpyridin-2-yl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,8-diazaspiro[4.5]decane
N-methyl-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
(1S,5R)-3-(1-benzofuran-2-ylmethyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)-2,6-difluorobenzamide
9-methoxy-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[3-(1,3-benzothiazol-2-yl)propanoyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
2-{2-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}acetamide
methyl 1-[(3R,5S)-1-[(4-chlorophenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-(2-{2-[(1-ethylpiperidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-(cyclopropylmethyl)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-N-methyl-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamido}-1-(pyrimidin-2-yl)pyrrolidine-2-carboxamide
1-{3-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
3-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-[(6-methylpyridin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2S)-2-amino-3-(1H-indol-3-yl)-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2,3-difluoro-4-methoxybenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
4-{[({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)amino]methyl}-1-methylpyrrolidin-2-one
6-(furan-3-yl)-2-{2-[(3-methoxypiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-[(2-hydroxyethyl)amino]-N-methylpyridine-3-carboxamide
1-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-3-propylurea
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-(2-ethylpyrimidin-5-yl)-6-fluoro-N-methyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
ethyl 4-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]piperidine-1-carboxylate
3-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
1-methyl-4-[3-oxo-3-(pyrrolidin-1-yl)propyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-chlorophenyl (7S,9aR)-8-methyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinolin-2-one
3-[3-({[4-(azepan-1-yl)butyl]amino}methyl)-1H-indol-1-yl]propanamide
[(6-methoxypyridin-3-yl)methyl](methyl)(oxan-4-ylmethyl)amine
3-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-[4-(5-methoxypyrimidin-2-yl)piperazin-1-yl]-1,3-benzothiazole