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3-[(2R,3R,6R)-5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]benzonitrile
(3R,4S)-4-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepan-1-yl)oxolan-3-ol
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
(1R,3S)-7-(7-chloro-4-methylquinolin-2-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-[2-(4-fluorophenyl)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
[(3R,4R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-pyrazole-3-carbonyl)piperidine
8-(5-chloropyridine-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(6-ethyl-2-methylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.5]decane
N,N-dimethyl-4-[3-(phenylamino)piperidine-1-carbonyl]piperidine-1-carboxamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
(1R,3s,6r,8S)-4-(4-ethylbenzoyl)-4-azatricyclo[4.3.1.13,8]undecane
[(2S,4R)-1-methyl-4-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}pyrrolidin-2-yl]methanol
N-ethyl-2-(4-fluoro-2-methoxyphenyl)-N-methylpyrimidin-4-amine
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
3-[3-(1H-imidazol-1-yl)propyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(N-methylmethanesulfonamido)ethyl]-2-phenylpyrimidine-5-carboxamide
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-[4-(trifluoromethoxy)benzenesulfonyl]piperidine
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-[3-(cyclohexyloxy)propyl]-3-(1H-pyrazol-4-yl)benzamide
2-(3-methoxyphenyl)-N-(oxan-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-(furan-2-ylmethyl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(prop-2-en-1-yl)acetamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyrrolidin-1-yl)benzamide
3-(1-benzyl-1H-pyrazol-5-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-({3-methyl-7-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
2-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrazine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1-methylcyclopropanecarbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclopentyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
2-{4-[3-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-1-yl}ethan-1-ol
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[3-(5-methylfuran-2-yl)phenyl]methyl}amine
2-(2-butoxy-4-fluorophenyl)-2-(morpholin-4-yl)acetic acid
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methoxypyridine-3-carbonitrile
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
N-methyl-2-[(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazol-4-yl)formamido]acetamide
2-[4-(benzylamino)butyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
methyl[(1-propyl-1H-imidazol-2-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]urea
2-chloro-N-(2-{[1-(methoxymethyl)cyclobutyl]formamido}ethyl)benzamide
3-(2,3-dihydroxypropyl)-3-methyl-1-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)urea
N,5-dimethyl-N-[(4-phenoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
6-methyl-N4-[1-(4-methylpyridin-2-yl)propyl]pyrimidine-2,4-diamine
3-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}pyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 6-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}pyridine-3-carboxylate