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3-{[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-cyclohexyl-N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-methyl-2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]thiophene-3-carboxamide
9-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-(1-{[benzyl(butyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
N,N-diethyl-1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)pyrrolidin-3-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(thiophen-3-yl)propanamide
2-methyl-6-[(5-methylhex-5-en-2-yl)amino]heptan-2-ol
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-ethyl-1,2,4-oxadiazole
3-({[(3,5-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-[2-(4-chloro-3-fluorophenyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
methyl 1-(2,7-dimethylquinoline-4-carbonyl)aziridine-2-carboxylate
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(methylsulfanyl)propanamide
methyl 4-[(5S,9aS,9bS)-2-(2-methoxyphenyl)-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]benzoate
1'-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-3H-spiro[2-benzofuran-1,4'-piperidine]-3-one
2-[(cyclopropylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[(2,4-dichlorophenyl)methyl]-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
4-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,3-dimethylpiperazin-2-one
[(2S,6S)-4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
[2-(2-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]dimethylamine
7-fluoro-3-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1-benzofuran-2-carboxamide
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-N-(thiophen-3-yl)piperidine-1-carboxamide
N-[(4-fluorophenyl)methyl]-2-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
N-[4-(3-methoxyphenyl)phenyl]-1-propanoylpyrrolidine-2-carboxamide
(1S,5R)-6-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-1-(oxolan-3-ylmethyl)urea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-carbamoylphenyl)methyl]pyrrolidine-3-carboxylic acid
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-phenoxybenzamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)propan-1-one
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(4-methylpyrimidine-5-carbonyl)piperidin-4-ol
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
2-[2-(3-propyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetic acid
3-hydroxy-N-methyl-N-[2-(oxan-2-yl)ethyl]pyridine-4-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(2-chlorobenzenesulfonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carboxamide
4-phenyl-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidine-4-carbonitrile
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-4-[2-oxo-2-(piperidin-1-yl)ethoxy]benzamide
2-hydroxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
3-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol
2-({6-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyrimidin-4-yl}amino)ethan-1-ol
(2S,4S)-4-amino-1-[(3,5-dimethoxyphenyl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
4-[(3S)-3-acetamidopyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
8-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one