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N-[2-(1H-imidazol-4-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
(3S,4R)-1-[2-(4-fluorophenoxy)ethanesulfonyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}-5-ethyl-1,2,4-oxadiazole
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}propanamide
9-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-(4-methoxy-2-methylphenyl)-1-(1,4-oxazepan-6-ylmethyl)urea
N-{[(3S,4S)-3-hydroxy-1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]methyl}-3-phenylpropanamide
3-[(3-methylpiperidin-1-yl)methyl]-N-(1,3-thiazol-2-yl)benzamide
1-cyclohexyl-N3-(2-methylpropyl)-N5-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3R,5S)-1-(2-methoxyacetyl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-indole-3-carboxamide
4-{furo[3,2-c]pyridin-4-yl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(1H-pyrazol-4-yl)benzamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
7-{[(1-hydroxybutan-2-yl)(thiophen-2-ylmethyl)amino]methyl}-4-methyl-2H-chromen-2-one
(2,1,3-benzothiadiazol-4-ylmethyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-[3-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenoxy)propyl]-1H-imidazole
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(4aS,8aR)-6-(pyridin-4-ylmethyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-2-(oxan-2-ylmethoxy)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-[4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperazin-1-yl]pyrazine
{2-[(isoquinolin-5-ylmethyl)[(3-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
4-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-fluoropyrimidin-4-yl)morpholine
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)piperazine-1-carboxamide
N-(1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
1-(2-chlorophenyl)-4-(7-fluoro-3-methyl-1H-indole-2-carbonyl)piperazin-2-one
1-[(4-fluorophenyl)methyl]-5-[(5-methyl-1H-pyrazol-1-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
3-{[(2-methoxyethyl)(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclohexyl-2-[1-cyclopropyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
6-{[5-(3-methoxypyrazin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5,6,7,8-tetrahydro-1,6-naphthyridine
5-[(2S)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(4-chlorophenyl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]butan-1-one
7-cyclopentyl-2-(3-hydroxypropyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazole
[(3,5-dichloropyridin-4-yl)methyl](ethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
4-[2-(3-methoxyphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
4-[4-(5-chloropyridine-3-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-(cyclopropylmethyl)-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
7-methyl-2-(pyridin-3-yl)-N-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine