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1-(furan-2-carbonyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-[({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenol
2,4-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-oxazole-5-carboxamide
N-cyclopentyl-5-(4-hydroxy-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1-benzofuran-2-carboxamide
({4-ethyl-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)thiomorpholine
2-(dimethylamino)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
1-[(2,6-difluorophenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
7-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(2-oxopyrrolidin-1-yl)-N-[2-(3-phenoxyphenyl)ethyl]propanamide
N-(1-methylpiperidin-4-yl)-2-(methylsulfanyl)-N-(pyridin-4-ylmethyl)acetamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(1,3-thiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(methoxymethyl)phenyl]-2-[4-(4-methoxyphenyl)piperazin-1-yl]acetic acid
N-({5-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
(1R,5R)-6-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
(3S,9aR)-3-[(benzyloxy)methyl]-8-(3-fluoro-4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-yl}morpholine
4-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-N-methyl-1,3-thiazol-2-amine
benzyl N-[1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]carbamate
N,N,4-trimethyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyrimidin-2-amine
2-{4-[(2-phenylphenyl)methyl]morpholin-3-yl}acetic acid
(1R,5R)-3-cyclobutanecarbonyl-6-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-3-propylurea
3-(1-propyl-1H-1,2,3,4-tetrazol-5-yl)-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[3-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-amine
N-{2-[bis(propan-2-yl)amino]ethyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-6-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
1-{3-oxo-3-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propyl}-1,2-dihydropyridin-2-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2,3-dimethoxyphenyl)-1H-imidazole
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
4-methoxy-2-(4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
4-(4-methylphenoxy)-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidine-4-carbonitrile
2-cyano-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-({7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-1-methylpiperidine-3-carboxamide
6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4-tert-butyl-1,2-dihydropyrimidin-2-one
ethyl 4-[(2-chlorophenyl)methyl]-1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxylate
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{5-[4-(dimethylamino)phenyl]-1H-indazol-1-yl}acetamide
2-{2-methyl-6-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}ethan-1-amine
1-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-5-phenylpentan-1-one
2-[(adamantan-1-ylmethyl)({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
4-(4-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]butanamide
3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-N-[(3-methylthiophen-2-yl)methyl]aniline
2-{5-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid