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1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(2-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
3-(1-butyl-3-phenyl-1H-1,2,4-triazol-5-yl)propanamide
(4aS,8aR)-6-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-hydroxy-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
8-(1-benzofuran-2-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}ethane-1-sulfonamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
4-[(4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}furan-2-yl)methyl]morpholine
(1R,5S,6S)-6-[(dimethylamino)methyl]-N-[3-(2-methylphenyl)phenyl]-3-azabicyclo[3.1.0]hexane-3-carboxamide
3-cyclohexyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
ethyl 1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
3-(3-fluorophenoxymethyl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
N,N-dimethyl-2-{[(2-methyloxan-2-yl)formamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
3-(3-hydroxy-3-methylbutyl)-N-(oxan-4-yl)benzamide
1-{3-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidine
N2-(4-methylpyridin-2-yl)-N1-(thian-4-yl)ethane-1,2-diamine
N-[(3,5-dimethoxyphenyl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-(1-methoxypropan-2-yl)acetamide
2-(4-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperidine-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)azetidine-1-carboxamide
6-(benzyloxy)-4-(furan-2-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
(1S,2S,9S)-11-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-(4-chlorobenzoyl)-1-(oxan-4-yl)piperidine
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]urea
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
2-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]acetic acid
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
1-[2-(1H-imidazol-4-yl)ethyl]-2-(oxolan-3-yl)-1H-imidazole
1-(4-methoxyphenyl)-4-[1-(pyridine-4-carbonyl)piperidin-3-yl]piperazine
N,1-dimethyl-N-[2-(phenylsulfanyl)ethyl]azepane-2-carboxamide
2-hydroxy-1-[4-(2-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-(1,3-benzothiazole-6-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1H-imidazol-2-yl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
1-({5-[(2-methoxy-3,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-cyclopropyl-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(1S,5R)-6-(cyclopropylmethyl)-3-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(2-methoxyphenyl)methyl]acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[3-(5-methylfuran-2-yl)butyl]amine