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(2S,4R)-4-amino-1-(1H-1,3-benzodiazole-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(1-cyclohexyl-4-hydroxypiperidin-4-yl)-N-(3,4-dimethoxyphenyl)-1-benzofuran-2-carboxamide
3-(ethylsulfanyl)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
N-[1-(pyrimidin-2-yl)piperidin-3-yl]azepane-1-sulfonamide
3-methoxy-6-[(E)-2-phenylethenyl]pyridazine
3-cyclopentyl-5-[(2-methylphenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
(1S,5R)-6-(3-fluoropyridine-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(3-methyloxetan-3-yl)methyl]acetamide
2-[3-(methoxymethyl)-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
(1R,2S)-1-{4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}-2,3-dihydro-1H-inden-2-ol
N-[2-(1H-imidazol-4-yl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-[(2-methoxynaphthalen-1-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
5-(4,8-dimethoxynaphthalen-1-yl)-1-ethyl-1H,4H-pyrazolo[3,4-d]imidazole
4-[4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepane-1-carbonyl]oxane-4-carbonitrile
(1S,6R)-9-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-({7-[2-(5-fluoro-2-methylphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)propanamide
5-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
7-(3,6-dimethylpyrazin-2-yl)-4-(oxolan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]isoquinoline
1-methyl-4-(quinoline-6-carbonyl)piperazin-2-one
8-chloro-2-methyl-N-[1-(methylcarbamoyl)cyclohexyl]quinoline-4-carboxamide
3-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
1,6-dimethyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
2-chloro-N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(4-fluoro-3-methylbenzoyl)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(oxan-2-ylmethyl)benzamide
3-{[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
1-cyclohexyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
2-{4-[(2E)-3-phenylprop-2-en-1-yl]morpholin-3-yl}acetic acid
N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrazin-2-amine
methyl 4-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)benzoate
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-(2-phenoxyethyl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
methyl 2-[cyclopentyl({[4-methoxy-3-(propan-2-yloxy)phenyl]methyl})sulfamoyl]benzoate
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-pyrazol-1-yl)butanamide
2-[5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)furan-2-yl]benzonitrile
1-(cyclohexylmethyl)-5-(morpholine-4-carbonyl)piperidin-2-one
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
2-{1-[(4-fluorophenyl)methyl]-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperazin-2-yl}ethan-1-ol
methyl (1R,3S,3aR,6aS)-5-ethyl-3-(2-methyl-1,3-thiazol-5-yl)-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
methyl 3-{[2-(4-chlorophenyl)acetamido]methyl}-5-(furan-2-amido)benzoate