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1-(cyclohexylmethyl)-N-cyclopropyl-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
4-ethyl-3-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(dimethylamino)ethyl]-8-(2-ethoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(benzyloxy)azetidine-1-carbonyl]-1-cyclopentylpiperidin-2-one
3-(azepane-1-carbonyl)-N-[(2-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1,4-dithiepan-6-amine
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-[2-(3-chlorophenyl)ethyl]-4-[(pyridin-4-ylmethyl)amino]pyrrolidin-2-one
8-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-[3,5-dimethyl-4-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
1-{[2-(1H-imidazol-2-yl)phenyl]methyl}-4-(pyridin-3-yl)piperazine
4-(1H-imidazol-1-ylmethyl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-methyl-1-[3-(morpholin-4-yl)propyl]-N-[2-(oxan-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-{1'-[(1-ethylpiperidin-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}pyridine-4-carboxamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-cyclopropyl-4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)quinoline
2-cyclopropyl-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methyl-N-(oxolan-2-ylmethyl)-1H-indazole-3-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl]methanol
3-hydroxy-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
N-methyl-4-oxo-4-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butanamide
3-methanesulfonyl-N-[(3R,4S)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]propanamide
8-[(2-chlorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
[(2S)-1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
7-[2-(3-chlorophenyl)-2-hydroxyacetyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 1-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}furan-3-carboxamide
2-amino-4-(2-chloro-4-hydroxyphenyl)-5-methyl-6-(pyridin-2-yl)pyridine-3-carbonitrile
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)-N-methylacetamide
1-[(3-fluorophenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-[(2-methoxyphenyl)methyl]acetamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}quinoline-6-carboxamide
9-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(furan-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-(3-hydroxy-2,2-dimethylpropyl)-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-2-methoxypyridine-3-carboxamide
2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-4-carboxamide
2,5-dioxo-6-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
7-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-oxa-7-azaspiro[4.5]decane
N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-(1H-pyrazol-4-yl)pyridine
N-[2-(3-chlorophenyl)ethyl]-1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carboxamide
(1-{[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol