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(1S,5R)-3-[2-(3-methoxyphenoxy)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-amino-1,3-thiazol-4-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
ethyl[2-(4-methanesulfonylphenoxy)hex-5-en-1-yl]methylamine
1-acetyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]piperidine-4-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
5-cyclobutanecarbonyl-1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3-{[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrazine-2-carboxamide
methyl 6-[3-(2-methylphenyl)piperidin-1-yl]pyrimidine-4-carboxylate
N4-{2-[(4-chlorophenyl)methoxy]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-[3-(methylcarbamoyl)phenyl]acetic acid
7-(cyclopropylmethyl)-2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
(2R,6R)-4-(isoquinoline-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[(4aS,8aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
methyl 4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-(2-methoxyethyl)-1-(1H-pyrazole-3-carbonyl)piperidine-3-carboxylic acid
N-(2,2-diphenylethyl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-(4-fluoro-3-methoxyphenyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
2-{4-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]piperazin-1-yl}-N,N-dimethylacetamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
({4-[1-(1H-indole-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
2-chloro-6-methoxy-4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
4-(2,5-dihydro-1H-pyrrole-2-carbonyl)-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1'-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
2-methyl-6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-(3-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
N-butyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-cyano-5-fluoro-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
5-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(dimethylamino)propanamide
4-[2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
5-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}pentan-1-amine
(4aR,7aS)-N,N-dimethyl-4-(5-methylpyrazine-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(4aS,8aS)-2-[(5-chloro-2,4-dimethoxyphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(1H-pyrrole-2-carbonyl)piperazine
(3R,9R)-11-(2-methoxybenzoyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
4-(propan-2-yl)-6-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
4-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-N-phenylpiperidine-1-carboxamide
3-hydroxy-S-[2-(2-hydroxyacetyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]butane-1-sulfonamido
1-ethyl-5-methyl-4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H-pyrazolo[3,4-d]imidazol-5-yl)-1H-pyrazole
(2S,4R)-1-[4-(4-fluorophenyl)-4-oxobutanoyl]-4-(2-hydroxyacetamido)-N-methylpyrrolidine-2-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
1-(2-{1-[(4-fluorophenyl)methanesulfonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
(1R,7S)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 1-[2-(dimethylamino)ethyl]-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate