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N-cyclopentyl-1-(2-methylpropyl)-5-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(3-fluoropyridin-4-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
(3S,4R)-1-(4-hydroxybenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-{2-[4-(isoquinolin-1-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)methanol
2-{3-[(E)-2-phenylethenyl]phenoxy}propanamide
7-[2-(3-phenylpyrrolidin-1-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-(3-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
2-(1-benzyl-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-{3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylfuran-2-carboxamide
N-(1-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
1-[2-(dimethylamino)ethyl]-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-2-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
6-{1-[(6-methoxy-1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
(3S,9aR)-3-(4-aminobutyl)-8-[(2-fluoro-5-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)thiophene-2-sulfonamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)piperidin-2-one
N-cyclopropyl-3-[5-(4-methylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N4-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
(3aR,6aR)-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-cyclopentylpropyl)-1-cyclopropyl-N-methyl-6-oxopiperidine-3-carboxamide
N-[(5-{3-cyclobutyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}furan-2-yl)methyl]-N-methylmethanesulfonamide
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-2-(1H-imidazol-1-yl)ethan-1-one
(1R,5S)-6-methyl-3-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-methoxypropyl)-8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
6-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
4-chloro-1-methyl-N-[3-(2-phenylacetamido)phenyl]-1H-pyrazole-3-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(pyrimidin-2-ylmethyl)piperidine-2-carboxamide
5-[(dimethylsulfamoyl)amino]-N-[2-(1H-indol-3-yl)ethyl]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
3-{2-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1-{5-[(3Z)-hex-3-en-1-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4-(2-methoxyethyl)-4H-1,2,4-triazole
1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-4-(4-ethylphenyl)butan-1-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
1-(3-methoxyphenyl)-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazin-2-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-methylbut-2-enoyl)piperidin-4-yl]oxy}benzamide
2,7-dimethyl-N-[2-(pyridin-3-yloxy)propyl]imidazo[1,2-a]pyridine-3-carboxamide
2-[(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3,5,7-trimethyl-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-indole-2-carboxamide
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]azepane
1-[(3-fluorophenyl)methyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
1-(3-ethylpiperazin-1-yl)-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-methoxyethyl)piperazine