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2-(5-acetylthiophen-3-yl)-1-[4-(benzyloxy)piperidin-1-yl]ethan-1-one
7-(cyclopropylmethyl)-2-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridin-3-ylmethyl)piperidin-3-yl]piperazine
5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-3-propyl-1,2,4-oxadiazole
2-phenoxy-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}urea
5-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-[ethyl(1,3-thiazol-4-ylmethyl)amino]-1λ6-thiolane-1,1-dione
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(3-fluoro-4-methylphenyl)methyl]pyrrolidin-2-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxopiperidin-1-yl)propanamide
4-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-[2-(azepan-1-yl)-2-phenylethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-{1-[(4-chlorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-2-ethylpyrimidine
N-cyclopropyl-1-[(1s,4s)-4-benzenesulfonamidocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
8-chloro-2-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
methyl({[5-(oxolan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})(thiophen-3-ylmethyl)amine
1-(4-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-imidazole
N-[(4-fluorophenyl)methyl]-3-(piperazine-1-carbonyl)aniline
6-methyl-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-chloro-5-acetamido-N-(1-fluoro-3-phenylpropan-2-yl)benzamide
1-(3-hydroxyazetidin-1-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-(3-methylbutyl)-2,4-dioxo-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
methyl 5-(2,6-dimethoxypyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-amino-3-ethyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-ethyl-4-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperazine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(4-methoxyphenyl)propyl]benzamide
2-[2-(3-fluorophenyl)-4-methylphenoxy]acetamide
({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyrimidin-2-amine
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(thian-4-yl)piperazine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(pyridin-4-ylmethyl)piperidin-1-yl]pyrimidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-[(2S)-1-hydroxypropan-2-yl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-methyl-5-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
3-(1,5-dimethyl-1H-pyrazol-4-yl)-4-[2-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(pyridin-2-ylmethyl)-4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]pyridine-2-carboxamide
(2S,4S)-4-amino-1-{2-[methyl(phenyl)amino]acetyl}pyrrolidine-2-carboxylic acid
4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}-1-(2-phenylethyl)piperidine
9-(4-methanesulfonylbenzenesulfonyl)-3-methyl-3,9-diazaspiro[5.6]dodecane
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
3-(4-methylphenyl)-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
2-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}benzoic acid
methyl 2-[1-(5-acetyl-4-methylpyrimidin-2-yl)pyrrolidin-3-yl]acetate
N-[1-(2-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-2-fluorobenzamide
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(2-methyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide