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1-[3-(azepane-1-carbonyl)phenyl]-3-[(1R,2S)-2-phenylcyclopropyl]urea
1-(4-chlorophenyl)-N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
(3R,5S)-N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(5S,9aS,9bS)-5-(4-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 2-{[2-(3-fluorophenyl)ethyl]sulfamoyl}-6-(1,2-oxazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(quinoline-4-carbonyl)pyrrolidin-3-yl]methanol
8-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(2,3-dihydro-1H-indene-1-carbonyl)-1-oxa-7-azaspiro[3.5]nonane
N-[2-(1H-imidazol-1-yl)ethyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-methyl-1,3-thiazol-2-amine
[(3R,4S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-{4-[2-(2-fluorophenyl)-1-(N-methyl-1-thiophen-2-ylformamido)ethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
(3R,4R)-4-(azepan-1-yl)-1-(quinolin-4-yl)piperidin-3-ol
5-(4-acetylphenoxymethyl)-N-[(2-amino-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
(1S,6R)-3-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-pyrazole-5-carboxamide
2-methyl-2-{4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]phenyl}propanenitrile
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1-methylpiperidin-4-yl)acetamide
4-({2-[(2-chlorophenyl)formamido]ethyl}amino)pyrimidine-5-carboxylic acid
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine-1-sulfonamide
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[2-(4-chloro-1H-pyrazol-1-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetamide
N-(4-methoxyphenyl)-1-[2-(2-methylpropanamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
1-{4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-[2-(dimethylamino)ethyl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxamide
6-(4-ethylphenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N,4-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-5-carboxamide
1-(furan-3-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
6-ethyl-5-methyl-N4-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide
4-{[3-(3-methoxypyrazin-2-yl)phenyl]methyl}morpholine
(1S,5R)-6-benzyl-3-(2-butoxyacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-3-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyridine-3-carboxylic acid
1-cyclohexyl-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methoxyphenol
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-indol-3-ylmethyl)piperidin-3-yl]propanamide
5-(morpholin-4-ylmethyl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-3-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-methyl-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazolidin-2-one
1-{4-[3-({[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one