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4-[(dimethylamino)methyl]-1-[(3-methylthiophen-2-yl)sulfonyl]azepan-4-ol
3-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinoxalin-2-one
1-(furan-2-carbonyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
1-[1'-(2,6-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-methyl-3-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(3-fluoropyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,1,3-trimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl](3-methylphenyl)methyl}dimethylamine
ethyl 2-(1-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazol-5-yl}-N-methylformamido)acetate
N-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
2-cyclopropyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane
4-methoxy-N-{2-[7-(3-phenylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
1-(5-methanesulfonamido-2-methylphenyl)-3-methyl-3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]urea
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3,9-diazaspiro[5.6]dodecane
3-(2-methoxyethyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylic acid
2-(2-aminoacetyl)-N-benzyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[3-(4-fluorophenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]azetidin-3-yl}pyridine
4-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}morpholine
2-{2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
1-(3,4-difluorobenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-{methyl[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
N-cyclopropyl-2-methyl-N-(thiophen-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[1-(3,5-dimethylbenzoyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
3-[2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(trifluoromethyl)benzamide
2-{4-[(3-ethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{[3-(2-phenylethyl)piperidin-1-yl]sulfonyl}pyridine
N-[(3S,4R)-1-[(3-methylquinoxalin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
N-[(2-phenoxypyridin-3-yl)methyl]-2-(propan-2-yl)pyrimidine-4-carboxamide
N-ethyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)phenyl]-3-methyl-4,5-dihydro-1H-pyrazol-5-one
2-methoxy-N-{1-methyl-2-phenyl-5-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}acetamide
4-(2-methoxyphenyl)-2-methyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
2-[methyl({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
N-(2-hydroxyethyl)-3,4,7-trimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-indole-2-carboxamide
4-[1-(5-propylpyrimidin-4-yl)pyrrolidin-3-yl]benzoic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5-methylpyrimidin-2-amine
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
1-[(3-methoxyphenyl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
N,5-dimethyl-1-[(methylcarbamoyl)methyl]-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide