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(2R,6S)-4-(5-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-2,6-dimethylmorpholine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
5-benzyl-N-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(butan-2-yl)-3-ethoxy-N-(pyridin-4-ylmethyl)propanamide
8-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
2-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
2-[3-(1H-imidazol-1-yl)propyl]-9-(pyrrolidine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
1-[4-(propan-2-yl)phenyl]-4-(thiomorpholine-4-carbonyl)pyrrolidin-2-one
N,N-dimethyl-1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
1-[2-methoxy-5-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-ethyl-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(4aR,8aS)-1-[2-(2-methylphenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-(pyridin-3-yl)propan-1-one
1-[(2-methylpyrimidin-5-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(3-chlorophenyl)-4-[2-(2-methoxyethoxy)acetyl]piperazin-2-one
8-(pyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-1H-1,3-benzodiazole-2-carboxamide
3-methoxy-6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridazine
1-benzyl-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
3-hydroxy-S-{2-[2-(methylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}butane-1-sulfonamido
5-(3-fluorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2,4-triazin-3-amine
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-methanesulfonyl-1,4-diazepane
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N-{4-[2-(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethoxy]phenyl}propanamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-hydroxy-5-methoxybenzamide
5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
(3S,4R)-1-[4-(4-methoxyphenyl)-4-oxobutanoyl]-4-phenylpyrrolidine-3-carboxylic acid
1-{4-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-4-oxobutyl}piperidin-2-one
(4aR,7aS)-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-(hydroxymethyl)-N-[(4-methoxypyridin-2-yl)methyl]pyridine-2-carboxamide
(benzylsulfamoyl)({[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl})amine
methyl (2S,4R)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
5-methyl-N-[2-(pyridin-3-yl)ethyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-tert-butyl-2-methyl-3-(4-methyl-2-oxopentanamido)benzamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(3-phenylpyrrolidin-1-yl)acetamide
1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
5,7-dimethyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
3-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
(1-{3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)(thiophen-2-yl)methanol
6-methyl-N-({1-[(4-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-2-carboxamide
2-chloro-N-(2-{3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}ethyl)benzamide
N-{[5-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide