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methyl (1S,3S,3aR,6aS)-3-(2-fluoro-6-methoxyphenyl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
3-chloro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(2R,6R)-4-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-1,6-dihydropyridine-2-carboxamide
methyl (2S,4R)-1-[(4-chlorophenyl)methyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxylate
2-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]amino}methyl)-5,8-dimethylquinolin-4-ol
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
(1R,5S,8R)-3-[(5-chlorofuran-2-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
N-(2-chlorophenyl)-3-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}propanamide
2-methyl-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
4-{2-[1-(5-fluoro-2-methylphenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholine
(3aR,6aR)-2-acetyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N2,N2-dimethyl-N4-[1-(thiophen-2-yl)butyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-(4-methyl-1H-pyrazol-1-yl)-1-[3-(3-methylphenoxy)azetidin-1-yl]propan-1-one
5-[(2-hydroxy-2-phenylethyl)(methyl)amino]-1-[2-(piperidin-1-yl)ethyl]azepan-2-one
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-benzyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
(5-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}furan-2-yl)methanol
3-{[(furan-2-ylmethyl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
3-({[(2,3-dimethoxyphenyl)methyl]amino}methyl)-7-methoxy-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
N-[2-({2-methyl-2,8-diazaspiro[4.5]decan-3-yl}formamido)ethyl]pyridine-3-carboxamide
N-ethyl-N-[(4-fluorophenyl)methyl]-3-(1H-pyrazol-4-yl)benzamide
1-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-phenylprop-2-yn-1-one
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(2-methoxyethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(pyridin-4-ylmethyl)-N-(4-sulfamoylphenyl)-1,4-diazepane-1-carboxamide
6-ethyl-4-[4-(2-phenoxyacetyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(2-methylpyridine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[5-(1-cycloheptyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
4-amino-5-(1-ethyl-1H-1,2,4-triazol-5-yl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
N-(1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
1-[1'-(5-chloropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-methyl-2-[2-(oxolan-2-ylmethyl)phenoxy]acetamide
N-[(5-chloro-1H-indol-2-yl)methyl]-4-(piperidin-1-yl)butanamide
5-[4-(trifluoromethyl)phenyl]pyrazin-2-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-2-carboxamide
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(1,3-thiazol-2-yl)propyl]acetamide
8-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(3-phenylpropyl)propanamide
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-7-(2-methylbenzoyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carbonitrile
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
N,N-diethyl-1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-sulfonamide
2,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
1-methyl-4-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S,4R)-4-amino-N-ethyl-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]pyrrolidine-2-carboxamide