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1-(2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-{3-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]phenyl}ethan-1-one
(3R,5S)-N3-[2-(5-methylfuran-2-yl)ethyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
N3-(1-benzothiophen-2-ylmethyl)-1-benzyl-N5-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
7-[2-(2,4-dimethoxyphenyl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
[7-fluoro-5-(2-methyl-1H-imidazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-cyclopropyl-1-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{3-[(1R,5S)-3-azabicyclo[3.3.1]nonane-3-carbonyl]phenyl}-2-methylbutan-2-ol
N-methyl-N-(3-phenoxypropyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
2-hydroxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
7-(3-chlorophenyl)-4-(furan-2-carbonyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-methylpyrimidin-2-yl)phenol
3-(3-aminopyrrolidine-1-carbonyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzene-1-sulfonamide
2-(dimethyl-1,2-oxazol-4-yl)-1-(7-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
methyl 4-[4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
1-(4-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
5-{2-[4-(3-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
methyl (2S)-2-{[(6,8-dimethyl-2-oxo-2H-chromen-4-yl)methyl]amino}-2-phenylacetate
N-[2-(4-methylpiperidin-1-yl)ethyl]-1,8-naphthyridine-2-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
5-(azepan-1-yl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-(cyclopropylmethyl)-4-(2,3-dimethoxyphenyl)-1H-pyrazole
1-{1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}piperidine-4-carboxamide
2-(2,5-dimethylphenoxy)-N-[(6-hydroxypyrimidin-4-yl)methyl]propanamide
9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[(2,4-dimethoxyphenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-phenyl-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
6-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(oxan-4-yl)pyrrolidin-3-ol
N,1-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 4-[5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
5-methyl-N-(3-{5-methyl-4-[(2-oxo-2-phenylacetamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
3-chloro-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
N-{1-cyclopentyl-7-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}benzamide
N2-(5-ethylpyrimidin-2-yl)-N1-(4-methylpyridin-2-yl)ethane-1,2-diamine
(4aS,8aS)-2-{[3-(3-methoxyphenyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
N-[2-(1-benzylpiperidin-2-yl)ethyl]acetamide
2-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}benzoic acid
5-(1-benzyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1H-imidazole-4-carboxylic acid
4-(1-methyl-1H-imidazol-2-yl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-4-carboxamide
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-cyclopropyl-5-[2-(pyridin-2-ylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide