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2-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-6-(4H-1,2,4-triazol-4-yl)pyridine
N-[(2,3-difluorophenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
7-fluoro-3-({methyl[3-(phenylsulfanyl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
N,1,3-trimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-benzyl-1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
N-(oxolan-3-yl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-(3-acetyl-1H-pyrazole-5-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
2-amino-6-cyclopropanecarbonyl-4-(3-methyl-1H-indol-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,4R)-N,N-dimethyl-1-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]-4-(propan-2-yl)pyrrolidin-3-amine
methyl 4-(5-methyl-4-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
(2-fluoro-5-{thieno[2,3-d]pyrimidin-4-yl}phenyl)methanol
1-cyclohexyl-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane
(4aR,7aS)-1-benzyl-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2-chloro-6-fluorophenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2,6-dioxo-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl (1S,3S,3aR,6aS)-3-(1-ethyl-1H-pyrazol-4-yl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
methyl 1-{2-hydroxy-3-[3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(4-fluorophenoxymethyl)piperidine
6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(2S)-2-amino-1-[4-(4-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
6-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-3-yl)propanamide
ethyl 1-(1-{4-[(1-phenylethyl)carbamoyl]phenyl}piperidin-4-yl)piperidine-4-carboxylate
N-(1-hydroxybutan-2-yl)-4-oxo-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
5-methanesulfonyl-4-(piperidin-3-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
1-cyclohexyl-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
2-[3-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
4-(piperidin-1-ylmethyl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}benzamide
({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)[1-(4-methoxyphenyl)ethyl]methylamine
6-(aminomethyl)-2-[3-({cyclopropyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-(3-methoxyphenyl)-1,2,4-triazin-3-amine
N,N-dimethyl-5-{1-[2-(pyridin-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
N-[2-(4-fluorophenyl)-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
7-(2-methylphenyl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
1-(thiophen-2-ylmethyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane
2-[1-(3-methylbut-2-en-1-yl)-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(4-fluorophenyl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)morpholine
1-(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-3-yl)ethan-1-one
1-(4-chloro-2-methylbenzoyl)-4-cyclopentyl-1,4-diazepane
(3S,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide