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6-methyl-2-({[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]amino}methyl)quinolin-4-ol
1-[(3-fluorophenyl)methyl]-4-{[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}pyrrolidin-2-one
5-[({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
4-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)piperazin-2-one
4-[5-(5-methyl-1-benzofuran-2-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
1-[(1S,5R)-6-[4-(diethylamino)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N,N-dimethyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazine-1-sulfonamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
4-{1-[4-(hydroxymethyl)phenyl]-1H-imidazol-2-yl}-2,6-dimethylphenol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
4-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]benzonitrile
2-[2-(3-phenyl-1,2-oxazole-5-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
1-(4-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
1-ethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-phenylacetamide
2-[5-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-[4-(benzyloxy)piperidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(adamantan-1-yl)-4-hydroxy-N-[(1S,2S)-2-hydroxycyclohexyl]pyrimidine-5-carboxamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(4-methoxyphenyl)furan-2-carboxamide
1-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]pyrrolidin-2-one
(3aS,6aS)-2-[(2,3-dichlorophenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3-oxopiperazin-1-yl)methyl]-N-(quinolin-6-yl)benzamide
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methanol
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(piperidine-1-carbonyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
1-[3-(aminomethyl)phenyl]-3-{1-[(2-methylphenyl)methyl]cyclopropyl}urea
3,5-dimethyl-4-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
dimethyl({[(1R,5S,6S)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-methyl-3-[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(but-3-yn-1-yloxy)-4-(4-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3S,4S)-1-[(3-chloropyridin-4-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
N-(furan-3-ylmethyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
{1-[4-(4-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
1-methyl-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazine-2-carboxylic acid
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidine-3-carboxylic acid
2-(4-fluorophenoxy)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(azepane-1-carbonyl)-N-(cyclopropylmethyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide