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1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-3-carboxamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(2-methylpyridin-4-yl)piperazine
4-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(3-methoxyphenyl)ethyl]benzamide
2-[(4-methoxyphenyl)methyl]-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-benzoxazole-6-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]acetamide
(3E)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]hex-3-en-1-one
N-(4-{[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]methyl}phenyl)acetamide
3-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-amino-N-methyl-N-[(4-phenoxyphenyl)methyl]pyridine-4-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
N-[(2-chloropyridin-3-yl)methyl]-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
3-hydroxy-3-({[(4-methylpyridin-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
2-(4-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}phenoxy)acetic acid
3-[1-(2-amino-2-methylpropanoyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
[2-(dimethyl-1,3-thiazol-2-yl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]acetamide
1-(diethylamino)-3-[2-methoxy-4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(dimethyl-1,3-thiazol-4-yl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]acetamide
(3aR,6aR)-2-cyclopentyl-5-[(4-acetamidophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{4-[1-(quinolin-3-yl)-1H-imidazol-2-yl]phenyl}but-3-yn-1-ol
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-{2-[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
2-methoxy-1-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-1-yl)ethan-1-one
4-ethyl-3-{1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(4-methoxyphenoxy)propyl]-N-methyl-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-(2-methoxyethyl)-N-methyl-5-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrrolidine-3-carboxamide
N-{3-[5-(morpholine-4-carbonyl)furan-2-yl]phenyl}acetamide
(3aR,6aS)-5-(2-amino-5-methylpyrimidin-4-yl)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
(3S,4S)-1-[(3-chloropyridin-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-({3-[(3S)-3-ethylmorpholine-4-carbonyl]phenyl}methyl)azepane
1-(3-chloropyridin-2-yl)-3-(hydroxymethyl)piperidin-3-ol
1-cyclohexyl-4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[(3aS,6aS)-2-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
(3S,4S)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
2-(2-aminoethyl)-N-cyclopropyl-N-[(2-methoxyphenyl)methyl]quinazolin-4-amine
1-ethoxy-3-({2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
methyl({5-[(2R)-oxolane-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
2-[2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
N-[2-(azepan-1-yl)ethyl]-1-cyclopentyl-N-methyl-6-oxopiperidine-3-carboxamide
5-(2,3-dihydro-1-benzofuran-5-yl)-1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N'-(2-tert-butylphenyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)butanediamide
4-[(3-chloro-4-hydroxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(4S,4aS,8aR)-1-(3-amino-1H-1,2,4-triazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol