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(3R,4R)-3-cyclobutyl-4-methyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
5-benzyl-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
3-[5-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(pyridin-2-ylsulfanyl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
5-benzyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-[(8-chloroquinolin-2-yl)methyl]-N,N-dimethylpyrrolidin-3-amine
N-cyclopentyl-6-(4-cyclopentylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-({2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[(2-chlorophenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(2-methoxyphenyl)-N-[1-(methylcarbamoyl)cyclohexyl]-1H-pyrazole-4-carboxamide
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
1-ethyl-5-[1-(2-phenoxyethyl)-1H-imidazol-2-yl]-1H-1,2,4-triazole
1-({1-[6-(morpholin-4-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-phenylbutanamide
cyclohexyl({4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
8-(2,6-dimethylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({2-[(pyridin-3-yl)amino]ethyl}amino)pyrimidine-5-carboxylic acid
3-(2-methylpropyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2-oxazole-5-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-methyl-1H-imidazole-5-carboxamide
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}furan-2-carboxamide
ethyl 1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-methyl-N-{[5-({methyl[2-(pyridin-4-yl)ethyl]amino}methyl)furan-2-yl]methyl}methanesulfonamide
4-{1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl}benzoic acid
4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
4-(2-methylpyrrolidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{4-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2-chloro-6-fluorophenyl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,5S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
5-ethyl-3-{2-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
(4aS,8aS)-2-[2-(propan-2-yl)pyrimidine-4-carbonyl]-decahydro-2,7-naphthyridin-4a-ol
N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]butanamide
1'-(5-hydroxypyrazine-2-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(ethoxymethyl)pyrrolidine
N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-2-[(2,4-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
({4-[2-(dimethylamino)ethoxy]phenyl}methyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
4-(3-chloro-2-methylbenzenesulfonyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[4-(oxolan-2-yl)butyl]acetamide
4-(4-methoxybutyl)-N-(quinolin-6-yl)piperazine-1-carboxamide
3,5-di-tert-butyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(propan-2-yl)piperazine