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8-acetyl-2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(3-fluoropyridin-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
2-(5-acetylthiophen-3-yl)-1-[(3S,4S)-3-hydroxy-4-(thiomorpholin-4-yl)pyrrolidin-1-yl]ethan-1-one
2-methoxy-5-(5-methylpyridin-2-yl)pyridine
(1S,5R)-3-methyl-6-[3-methyl-4-(morpholin-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
9-[4-(1H-imidazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-(3-fluorophenyl)-N'-[(1-methylpiperidin-3-yl)methyl]butanediamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(oxolane-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(3R,4R)-1-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
1-(4-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-(3-methyl-3-phenylpiperidine-1-carbonyl)-1λ6-thiane-1,1-dione
(4aS,7aR)-4-[(4-ethoxyphenyl)methyl]-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
8-(3-methylbut-2-en-1-yl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methylphenol
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(2S)-1-hydroxypropan-2-yl]benzamide
(1S,6R)-9-[2-oxo-7-(propan-2-yloxy)-2H-chromene-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-methyl-2-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-3,4-dihydro-2H-1,4-benzoxazine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1-methyl-1H-pyrazole
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
3-[2-(oxolan-3-yl)ethyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
4-methyl-6-{4-[(morpholin-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-amine
1-(3-methoxybenzoyl)-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
4-(3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonyl}benzoyl)morpholine
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-2H-1,3-benzodioxole-5-carboxamide
2-benzyl-4-[(3,4-dimethoxyphenyl)methyl]morpholine
2,6-dimethyl-4-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenol
1-(2,3-dihydro-1H-inden-2-yl)-4-[(6-ethoxypyridin-3-yl)methyl]piperazine
1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-{2-[(2-methylphenyl)carbamoyl]acetyl}piperidine-4-carboxylic acid
2-{4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(1S,5R)-3-[4-(4-fluorophenyl)-4-oxobutyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(3,4-dimethoxyphenyl)-9-methoxy-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,5S)-1-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)quinolin-8-ol
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-(3-chloro-4-methylbenzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
4-ethyl-2-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,3-thiazole
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
6-[1-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-[(3S)-1-benzylpyrrolidin-3-yl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole