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N-[(2-methoxyphenyl)methyl]-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
1-(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)ethan-1-ol
2-(dimethylamino)-2-(2-methylphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
(1R,5S,8S)-8-methoxy-3-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3-azabicyclo[3.2.1]octane
8-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,2,3,6-tetramethyl-N-(thian-4-yl)quinoline-4-carboxamide
N-(3,3-diphenylpropyl)-2-(morpholin-2-yl)acetamide
methyl (2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(2-methylquinoline-4-amido)pyrrolidine-2-carboxylate
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
N-(3-cyclopentylpropyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-(2-methoxyethyl)-3-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
[(3-chloro-4-fluorophenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(1,3-thiazol-2-yl)piperidine
3-acetamido-N-[2-(propylsulfanyl)phenyl]pyrrolidine-1-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
methyl[(4-methyl-1H-imidazol-5-yl)methyl](quinolin-5-ylmethyl)amine
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
5-(3-fluorophenyl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
1-(5-fluoro-2-methoxyphenyl)-3-[2-(propylsulfanyl)ethyl]urea
methyl (2S,4R)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxylate
(3R,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]pyrrolidin-3-amine
5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-imidazole
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1-(pyrimidin-2-yl)piperidin-4-amine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopentylacetamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidine-4-carboxamide
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N,N-dimethylacetamide
1-(furan-2-carbonyl)-4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
2-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}pyridine-4-carboxamide
(2S,4R)-1-benzyl-N-(2-methoxyethyl)-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
4-acetamido-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}benzamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-(2,4-dimethoxybenzoyl)-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
[(4,5-dimethylfuran-2-yl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(4aR,7aS)-1-acetyl-4-[(4-fluoro-3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2-hydroxyethyl)(methyl)amino]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
(3S,9aR)-8-[(4-methoxyphenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-(2-phenylethyl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
4-(3-fluorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
1-cycloheptyl-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
(8R,9aS)-8-hydroxy-2-{[1-(phenoxymethyl)cyclopropyl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione