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2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)propanamide
2-cyclopentyl-N-[3-(4-{[2-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)phenyl]acetamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(2-methyl-1H-indol-3-yl)acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
4-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-5,6-dimethylpyrimidine
(2S,4R)-4-[3-(2-amino-1,3-thiazol-4-yl)propanamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
methyl 3-[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]propanoate
5-ethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N3-[3-(1H-1,3-benzodiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
3-ethyl-N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
2,3,6-trifluoro-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-{4-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}-4,6-dimethylpyrimidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-amino-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
5-methoxy-1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-indole-2-carboxamide
1-(furan-3-carbonyl)-3-[2-(4-methoxyphenyl)ethyl]piperidine
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
6-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
2-{2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}-5,6-dimethyl-1H-1,3-benzodiazole
3,3,3-trifluoro-2-hydroxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)propanamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-cyclopropyl-9-(4-fluorobenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2-(pyridin-3-yl)quinoline
methyl 4-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-4-oxobutanoate
2-(2,4-dichlorophenoxy)-N-methyl-N-(thian-4-yl)acetamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(pyridin-3-yloxy)acetyl]-decahydro-1,6-naphthyridin-2-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
3-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
3-(2-fluorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]-3-phenylpropanamide
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[4-(pyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
N-[3-(1H-indol-2-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(1-propylpiperidin-4-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
7-({2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-4-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decane
5,5-dimethyl-1-({3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)imidazolidine-2,4-dione
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
2-methyl-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][2-(piperidin-1-yl)ethyl]amine
1-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-methoxy-1-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-indole-2-carboxamide
1-{1-[4-(furan-2-yl)phenyl]piperidin-4-yl}-1,2,3,6-tetrahydropyridine