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3-(5-{1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
3-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-benzoxazole
(3S)-1-[7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)acetamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)[(6-methylpyridin-2-yl)methyl]amine
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-[3-(methylsulfanyl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N2-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
(1S,5R)-6-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
7-(2-methoxyethyl)-2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-(3-fluorophenyl)-N-{[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
(1S,5R)-3-cyclobutanecarbonyl-N-[4-(propan-2-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
9-(but-3-yn-1-yloxy)-4-(3-methoxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 7-oxo-3-(2-phenoxyacetyl)-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-2-[methyl({[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl})amino]propanamide
N-{1-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-1-oxopentan-2-yl}acetamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
9-(3,4-difluorobenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(furan-3-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[3-(2-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]dimethylamine
4-(6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridazin-3-yl)thiomorpholine
2-[(1S,5R)-3-[(3-hydroxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(methylsulfanyl)-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
2-(6-aminopyridin-3-yl)-2-(azepan-1-yl)acetic acid
4-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)methyl]benzoic acid
1-(4-methoxyphenyl)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]cyclopentane-1-carboxamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(1H-indol-4-ylmethyl)methylamine
4-[({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-1,3-thiazol-2-amine
N-(2-phenylethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-4-carboxamide
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
1-{3-[3-(furan-3-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
3-[(2-aminopyridin-4-yl)methyl]-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-(2-methoxyphenoxy)-N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]azetidine-1-carboxamide
2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethan-1-ol
(2S,4S)-4-(2-chlorobenzamido)-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-propoxypiperidine
N-[(3S,4R)-1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
N-[(3-methoxyphenyl)methyl]-3-[1-(quinoline-6-carbonyl)piperidin-3-yl]propanamide
2-(morpholin-4-ylmethyl)-N-(4-oxo-4H-chromen-6-yl)piperidine-1-carboxamide
[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(furan-2-yl)ethyl]acetamide
4-[3-(methylsulfanyl)propyl]-2-(2-phenylethyl)morpholine
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(2-phenoxyethyl)piperazine
dimethyl[(4-methyl-5-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
[3-(2-methoxyethyl)-1-(1-phenylpiperidin-4-yl)piperidin-3-yl]methanol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide