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4-{2-[3-(2-methoxyethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
2-methoxy-1-[1'-(pyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-{2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(2-methoxyethyl)-1,3-dimethyl-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-{4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one
5-[2-(azocan-1-yl)acetyl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-cyclobutyl-6-methyl-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]pyrimidin-2-amine
4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(propylsulfamoyl)benzamide
[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
4-{2-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
1-(5-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)ethan-1-one
(3S,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(furan-3-ylmethyl)-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
1-(2-methoxyphenyl)-4-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]piperazin-2-one
8-{imidazo[1,2-a]pyridine-2-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-fluoro-5-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]-2-methylpropanamide
1-(2,3-dihydro-1H-inden-2-yl)-5-(1H-imidazol-4-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
N,N,3-trimethyl-2-[(trimethylpyrimidin-4-yl)amino]butanamide
2-(1H-imidazol-1-yl)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1-(4-methoxyphenyl)-6,6-dimethyl-N-[(3-methylquinoxalin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-hydroxy-1-{8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
4-methoxy-3-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-(4-chloro-2-fluorophenyl)-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-pentylbenzene-1-sulfonamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclopentyl-N5-[(2-methoxynaphthalen-1-yl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-methoxybenzoyl)-4-(3,3,4,4,4-pentafluorobutyl)piperazine
6,7-dimethoxy-2-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-methyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)pyrimidine
N-methyl-N-[(5-{[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-yl)methyl]methanesulfonamide
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
4-(6-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyrazine-2-carbonyl)morpholine
2-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)benzoic acid
1-(2-aminoethyl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
8-chloro-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}quinoline
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-{2-[2-(3-fluoro-2,4-dimethylphenyl)-1H-imidazol-1-yl]-1-(pyridin-2-yl)ethyl}morpholine
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
4-methyl-6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
2-(4-{[1-(cyclopropylmethyl)-7-oxoazepan-4-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
5-(1,3-benzothiazol-2-ylmethyl)-N-benzyl-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide