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(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-(naphthalen-1-ylmethyl)piperidine-3,5-dicarboxamide
N-(furan-2-ylmethyl)-3-{[1-(1H-indol-2-yl)ethyl](methyl)amino}propanamide
3-(3-hydroxy-3-methylbutyl)-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]benzamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
ethyl 1-(dimethyl-1,2-oxazole-4-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]methanesulfonamide
1-cyclopropyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
3,5-dichloro-4-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]benzamide
8-(4-hydroxybenzoyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
5-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
[2-(1H-indol-3-yl)ethyl](methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
(1R,5S,8S)-8-methoxy-3-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-3-azabicyclo[3.2.1]octane
5-methanesulfonyl-1'-(2-methylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-methyl-N-({1-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)but-2-enamide
9-methoxy-N-methyl-3-[2-(2-methylphenyl)acetyl]-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-chloro-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-pyrazol-5-amine
4,4-difluoro-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[4-(4-phenyl-1,3-thiazol-2-yl)piperazin-1-yl]methyl}benzonitrile
2-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
5-chloro-2-methyl-6-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrimidin-4-ol
1-{1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]ethyl}-4-methylpiperazine
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
(2S,4R)-4-amino-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-butyl-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
11-(4-ethylpiperazin-1-yl)-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(3-methoxyquinoxalin-2-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
2-amino-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-6-(propan-2-yl)pyrimidine-4-carboxamide
2-{4-[(dimethylamino)methyl]phenyl}-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
2-(5-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-(2-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
6-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
6-(cyclobutylamino)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
N-[(1R,2S)-2-phenylcyclohexyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-benzyl-6-(morpholine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-({3-[4-(piperidin-1-ylmethyl)phenyl]phenyl}methyl)morpholine
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-[1-(2-amino-6-hydroxypyrimidin-4-yl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
N-[3-(pyridin-2-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-(oxan-4-yl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
9-(1H-indol-5-ylmethyl)-3-oxa-9-azaspiro[5.5]undecane
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[2-(trifluoromethyl)benzoyl]-1,4-diazepan-6-yl}oxy)acetamide
4-hydroxy-N-[(5-methylfuran-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N3-butyl-1-cyclohexyl-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-benzyl-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one