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1-(4-acetylpiperazin-1-yl)-3-(4-methoxyphenyl)-3-phenylpropan-1-one
N-[1-(furan-2-yl)ethyl]-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
2-(5-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(2-oxopiperidin-3-yl)benzamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidine
methyl 5-oxo-5-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pentanoate
(1R,5R)-6-(2-methoxyethyl)-3-[1-(4-methylphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
methyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})(quinoxalin-2-ylmethyl)amine
2-benzyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-butyl-N-ethyl-3-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
ethyl 1-(2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetyl)piperidine-2-carboxylate
N-cyclopropyl-3-{[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]sulfamoyl}benzamide
4-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
4-(4-fluorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butanamide
2-[1-(2-methoxyphenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[2-(ethylcarbamoyl)phenyl]-N-propylpyridine-3-carboxamide
5-(3,4-dimethylphenoxymethyl)-3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazole
3-[2-hydroxy-2-(pyridin-3-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(3-chlorophenyl)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}piperidin-4-amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
N-methyl-1-(oxolan-2-ylmethyl)-N-[(4-phenoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(thiophene-2-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(morpholin-3-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
7-methyl-2-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-chloro-5-(2-methoxypyridin-3-yl)-N-methylbenzamide
methyl 3-cyclopropaneamido-6-({methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
(3R,4S)-4-[methyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amino]oxolan-3-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-2-one
2-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)benzonitrile
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}benzoic acid
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2,4-difluorophenyl)methyl]piperidine
2-oxo-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-[(2-chloro-6-fluorophenyl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7-methanesulfonyl-N,4-dimethylquinazolin-2-amine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
{1-[1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)piperidin-4-yl]ethyl}dimethylamine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(1H-imidazol-1-yl)acetamide
2-(2,3-dimethoxyphenyl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazole
N-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-methyloxan-4-amine
3-(2-ethoxypyridin-3-yl)pyridin-2-ol
2-(adamantan-1-yl)-4-hydroxy-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyrimidine-5-carboxamide
4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]sulfonyl}-3,5-dimethyl-1,2-oxazole
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylimidazo[1,2-a]pyrimidine-3-carboxamide