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6-fluoro-2-{[(thiolan-3-yl)amino]methyl}quinolin-4-ol
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[3-(1H-pyrazol-1-yl)propyl]amine
2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidine
1-[4-(dimethyl-1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2,2-diphenylethan-1-ol
1-[(4-fluorophenyl)methyl]-4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrrolidin-2-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
2-(3,4-dimethylphenoxy)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-cyclopentyl-6-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(2-chloro-4,6-dimethylphenyl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
4-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1,2,3,4-tetrahydroquinolin-2-one
N-(2-{[6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}ethyl)acetamide
2-(2,5-dimethylphenoxy)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
N-[2-(1H-imidazol-1-yl)propyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-{[4-(5-fluoro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
3-(3-fluorophenyl)-3-{2-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N,1-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-indole-3-carboxamide
(4aR,6R,8aS)-2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-(2-phenylethyl)-4-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,4-diazepan-1-yl)-1,3-benzothiazole
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
(1S,6R)-9-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-methyl-1H-pyrazol-1-yl)acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-({[4-(diethylamino)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(1,3-benzoxazol-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-(quinolin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
7-acetamido-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)furan-2-carboxamide
({1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
2-ethyl-4-[3-(1H-pyrazol-3-yl)phenyl]aniline
2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-N-(prop-2-en-1-yl)aniline
(2S,4R)-4-amino-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-(naphthalen-1-yl)-3-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanoic acid
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-phenylacetamide
1'-(7-methyl-1-benzofuran-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-propyl-5-[3-(trifluoromethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-[(3,4-dimethoxypyridin-2-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
methyl (2S,4R)-1-methyl-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-amido]pyrrolidine-2-carboxylate
4-benzyl-3-ethyl-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-1,4-diazepan-5-one
(3R,4R)-3,4-dimethyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-ol
2-({2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
6-[(3-fluorophenyl)methoxy]-4-(1-hydroxypropan-2-yl)-1-(2-phenylethyl)-1,4-diazepan-2-one
8-(2,7,8-trimethylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-phenyl-7-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(4-chlorophenyl)methyl]-8-(oxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
(2S)-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-propanoylpyrrolidine-2-carboxamide