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N-(1,3-dihydroxypropan-2-yl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
2-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-ol
{4-[(5-phenylthiophen-2-yl)methyl]morpholin-3-yl}methanol
3-cyclopropyl-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
4-[1-(5-acetylthiophene-3-carbonyl)piperidin-3-yl]benzoic acid
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-methoxybenzamide
(1S,5R)-6-(2H-1,3-benzodioxol-5-ylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethyl-1,3-thiazol-5-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
11-{[(2,4-difluorophenyl)methyl]amino}-4-[2-(morpholin-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-methylpyrimidin-2-amine
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(5-tert-butyl-1H-pyrazol-3-yl)pyridine-3-carbonitrile
2-{2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
5,6-dimethyl-3-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydropyridin-2-one
(3R,4S)-4-{ethyl[(5-ethylpyridin-2-yl)methyl]amino}oxolan-3-ol
5-(2-methyl-4-phenylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-[(2,5-dimethylphenyl)methyl]-1-phenylpiperazin-2-one
N2,N2,5,6-tetramethyl-N4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine
3-methyl-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
2-methyl-2-{4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazol-1-yl}propane-1,3-diol
2,3-dimethyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-methanesulfonylphenyl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-phenylpyridine-3-carboxylic acid
methyl 9-[3-(N-methylacetamido)pyrrolidin-1-yl]-3-azaspiro[5.5]undecane-3-carboxylate
2,2-dimethyl-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-ethyl-5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-propylquinoline-4-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]pyrazin-2-amine
N4-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
4-fluoro-2-[4-(1H-pyrazol-5-yl)phenyl]phenol
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
6-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}cyclopropane-1-carboxamide
2-methyl-6-(1H-pyrazol-3-yl)-4-(trifluoromethyl)pyridine
3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
[3-(1H-imidazol-1-yl)propyl]({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
3-(1H-1,3-benzodiazol-1-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(2-methylphenoxy)piperidine
1-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-[2-(dimethylamino)-4-methylpyrimidine-5-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
N-(furan-2-ylmethyl)-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-methyl-1,4-diazepan-1-yl)propan-1-one
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)pyrazine-2-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide