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6-(2-chlorophenyl)-N-(2-methoxyethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-(1H-imidazol-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
ethyl 1-(oxan-4-yl)-3-(2-phenylethyl)piperidine-3-carboxylate
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]pyridin-3-ol
2-[4-chloro-2-({methyl[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]acetic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
1-(3-methanesulfonamidophenyl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
8-[3-(2-methoxyphenoxy)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
(2R,4R)-N-(1-ethylpiperidin-4-yl)-4-hydroxy-N-[2-(pyridin-2-yl)ethyl]pyrrolidine-2-carboxamide
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
(3aS,6aS)-1-[(2-fluoro-5-methoxyphenyl)methyl]-5-(thiophene-3-carbonyl)-octahydropyrrolo[2,3-c]pyrrole
2-butyl-8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(furan-3-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
3-(5-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
(3R,4S)-4-[ethyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})amino]oxolan-3-ol
6-methyl-4-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
4-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]-N-[4-(2-hydroxyethyl)phenyl]benzamide
3-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanamide
2-(4-{8-oxo-2-oxa-7-azaspiro[4.5]decan-7-yl}piperidin-1-yl)pyridine-3-carbonitrile
4-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2,6-dimethyl-5-{[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
1-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
9-{[4-(2-aminoethyl)phenyl]methyl}-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(morpholine-4-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-propanamidobenzamide
1-(pyrazine-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(3-hydroxy-2,2-dimethylpropyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(2-amino-4-methyl-1,3-benzothiazol-6-yl)-5-oxopyrrolidine-3-carboxylic acid
3-cyclopropyl-4-(3,4-diethoxybenzoyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
ethyl 1-[(1,1-dioxo-1λ6-thiolan-3-yl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
4-(4-cyclobutanecarbonyl-2-oxopiperazin-1-yl)benzonitrile
1-[3-(methylsulfanyl)propyl]-4-phenyl-5-propyl-1H-imidazole
2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)-N-methylacetamide
5-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
2-(1H-imidazol-1-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}propanamide
2-ethyl-8-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-methyl-1,4-diazepan-1-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-N-[(2-methylphenyl)methyl]-7-azaspiro[3.5]nonane-7-carboxamide
3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-inden-1-one
2-benzyl-9-(5-ethyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-4-amine
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(piperidin-1-ylmethyl)piperidin-1-yl]propan-1-one
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
8-[3-(oxan-4-yl)-5-[(2R)-pyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl]quinoline
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylpropanamide