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(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyridazine-3-carbonyl)piperidin-3-ol
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyrazin-2-yl)ethyl]amine
3-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
2-amino-4-(1-methyl-1H-indol-6-yl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
1-(2-methylpropyl)-N-[2-(methylsulfanyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aR)-2-acetyl-5-({[2-(4-methoxyphenyl)ethyl]carbamoyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{2-[2-(methylsulfanyl)phenyl]ethyl}-1λ6-thiolane-1,1-dione
(3R,4R)-1-({3-[(4-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-4-(hydroxymethyl)piperidin-3-ol
5-(3-{1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
5-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
[(5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-3-yl)methyl]dimethylamine
2-[1-(3-methylbut-2-en-1-yl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
N-[(2,3-dimethoxyphenyl)methyl]-4-methyl-5-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})(oxolan-3-ylmethyl)amine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
2-(2-hydroxyethyl)-8-[5-(hydroxymethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(2-fluorophenyl)pyrrolidine
N-[(5-methylpyrazin-2-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
7-{2-[(2-phenylethyl)sulfanyl]pyridine-3-carbonyl}-2-oxa-7-azaspiro[4.5]decane
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
8-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-methyl-4-phenylpyridine-3-carboxamide
2-{[(3-ethoxyphenyl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})amino}ethan-1-ol
3-{[cyclohexyl(methyl)amino]methyl}-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-(butan-2-yl)-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
4-[(4-methoxyphenyl)methyl]-1-(3-methylbenzoyl)-1,4-diazepan-5-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(5-methyl-1H-indazole-3-carbonyl)piperidin-3-ol
N-[1-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
2-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}benzoic acid
N-ethyl-6-(2-hydroxyethyl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(4-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
1-[1-(4-fluorobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{5-[(4-benzoylpiperazin-1-yl)methyl]thiophen-2-yl}prop-2-yn-1-ol
(benzylsulfamoyl)({3-[(dimethylamino)methyl]phenyl}methyl)amine
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-4,6-dimethylpyridine-3-carbonitrile
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)propanamide
N,2-dimethyl-N-[2-phenyl-1-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]furan-3-carboxamide
2-[5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-(4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-(1-{[1-(3-methylpyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3-(2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
N-(5-chloro-2-methoxyphenyl)-3-(1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
N-methyl-N-(oxan-2-ylmethyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethan-1-one
2-({[5-(methoxymethyl)thiophen-2-yl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide