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1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
[1-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
(4aS,8aR)-6-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole
2-[(1S,5R)-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)oxolane-2-carboxamide
6-cyclopropyl-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]pyrimidin-4-amine
N-butyl-N-(4-hydroxybutyl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1,3-benzoxazole-6-carboxamide
N-(1-methyl-1H-1,2,3-triazol-4-yl)-2-(1H-pyrazol-1-yl)acetamide
(2R,3S,6R)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}piperidin-1-yl)-2-methoxyethan-1-one
N-(1H-indol-4-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)propanamide
1-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)(phenyl)methyl]-1H-1,2,3,4-tetrazole
3-{[butyl(methyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
ethyl 2-[4-(4-methoxybenzoyl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
2-[benzyl(methyl)amino]-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2,3-dihydro-1H-indene-2-carboxamide
(1R,9aR)-1-[4-(4H-1,2,4-triazol-4-yl)phenoxymethyl]-octahydro-1H-quinolizine
2-(7-methyl-1H-indol-3-yl)-N-(prop-2-en-1-yl)pyridine-3-carboxamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
2-chloro-5-acetamido-N-[2-(3-hydroxypiperidin-1-yl)ethyl]benzamide
N-{4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
4-phenyl-N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
1-ethyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(4-fluorophenyl)-2-[(5-methoxy-1-methyl-1H-indol-2-yl)formamido]propanoic acid
2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-4-({[3-(methylsulfanyl)phenyl]methyl}amino)pyrrolidin-2-one
4-hydroxy-1-[2-(3-methylphenyl)benzoyl]piperidine-4-carboxylic acid
2-(dimethylamino)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(4-methylphenyl)ethan-1-one
4-chloro-N-[(3R,5S)-1-cyclobutanecarbonyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N,N-dimethyl-2-{2-[({3-[(pyridin-3-yl)amino]propyl}carbamoyl)amino]phenyl}acetamide
3-chloro-N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
4-benzyl-7-(5-chloropyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(propan-2-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
(4aR,7aS)-1-{2-[ethyl(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
2-methoxy-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]quinoline
3-amino-1-(1-benzofuran-5-ylmethyl)pyrrolidine-3-carboxylic acid
8-[3-(ethylsulfanyl)propanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazole
3-methoxy-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-5-methoxyphenol
N,N-diethyl-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1,2,5-thiadiazole-3-carbonyl)piperidine